SCHEMBL27832141

SCHEMBL27832141

CC1C(=O)N(C(CC=O)C(=O)O)CCN1c1cccc(OC(F)(F)F)c1

nearest known ligand 0.42

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
NOTUM Q6P988 1/20 0.42
FFAR4 Q5NUL3 1/20 0.40
CHRM2 P08172 3/20 0.37
CHRM1 P11229 2/20 0.37
CHRM4 P08173 6/20 0.37
DRD2 P14416 3/20 0.37
DRD3 P35462 3/20 0.37
KCNH2 Q12809 3/20 0.37
MCHR1 Q99705 1/20 0.37
ACACB O00763 1/20 0.36
HCRTR1 O43613 1/20 0.35
HCRTR2 O43614 1/20 0.35
CCKBR P32239 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL734130 0.92 NOTUM (0.38) NOTUMFFAR4CHRM2CHRM1CHRM4
SCHEMBL27933836 0.87 NOTUM (0.45) NOTUMFFAR4CHRM2CHRM1CHRM4
SCHEMBL27832131 0.82 NOTUM (0.39) NOTUMFFAR4CHRM2CHRM1CHRM4
SCHEMBL733975 0.81 NOTUM (0.41) NOTUMFFAR4CHRM2CHRM1CHRM4
SCHEMBL27812001 0.80 NOTUM (0.43) NOTUMFFAR4CHRM2CHRM1CHRM4
SCHEMBL734643 0.79 HSD17B10 (0.44)
SCHEMBL736399 0.79 LIPE (0.39) NOTUMFFAR4CHRM2CHRM1CHRM4
SCHEMBL736398 0.79 LIPE (0.39) NOTUMFFAR4CHRM2CHRM1CHRM4
SCHEMBL734564 0.77 DRD2 (0.45) NOTUMFFAR4CHRM2CHRM1DRD2
SCHEMBL734524 0.75 NOTUM (0.36) NOTUMCHRM2CHRM1CHRM4MCHR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-102112451-A Diazepan and piperazine derivatives modulators of chemokine receptors HOFFMANN LA ROCHE 2011-06-29 CN disclosed