SCHEMBL27832147

SCHEMBL27832147

CC1C(C=O)NCCN1c1ccc(N)c(C(F)(F)F)c1

nearest known ligand 0.36

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
HTR2A P28223 3/20 0.36
HTR2C P28335 3/20 0.36
HTR2B P41595 3/20 0.36
AR P10275 15/20 0.34
ADAMTS5 Q9UNA0 1/20 0.31
FFAR4 Q5NUL3 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL27832139 0.86 NOTUM (0.41) ARADAMTS5
SCHEMBL27811999 0.84 NOTUM (0.41) HTR2AHTR2CHTR2BARADAMTS5
SCHEMBL27811988 0.82 SIRT6 (0.51) HTR2AHTR2CHTR2BAR
SCHEMBL27811989 0.79 ALDH1A1 (0.46) HTR2AHTR2CHTR2BAR
SCHEMBL735198 0.75 BCL2A1 (0.43) HTR2AHTR2CHTR2BARADAMTS5
SCHEMBL27832140 0.74 NOTUM (0.41) HTR2AHTR2CHTR2BFFAR4
SCHEMBL2567623 0.70 AR (0.56) AR
SCHEMBL2793351 0.70 AR (0.56) AR
SCHEMBL2975255 0.70 AR (0.56) AR
SCHEMBL2980700 0.69 AR (0.52) AR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-102112451-B Diazepan and piperazine derivatives modulators of chemokine receptors HOFFMANN LA ROCHE 2014-01-22 CN disclosed
CN-102112451-A Diazepan and piperazine derivatives modulators of chemokine receptors HOFFMANN LA ROCHE 2011-06-29 CN disclosed