SCHEMBL27834151

SCHEMBL27834151

O=C(CO)Oc1ccc(-n2ccnc2)cc1

nearest known ligand 0.55

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP3A4 P08684 6/20 0.53
BAZ2B Q9UIF8 1/20 0.53
CYP2D6 P10635 6/20 0.52
CYP2C9 P11712 5/20 0.52
CYP1A2 P05177 4/20 0.52
CYP2C19 P33261 3/20 0.52
CYP19A1 P11511 1/20 0.52
HTT P42858 1/20 0.52
ENPP2 Q13822 1/20 0.51
MKNK1 Q9BUB5 1/20 0.51
MKNK2 Q9HBH9 1/20 0.51
ADH5 P11766 1/20 0.50
CA1 P00915 2/20 0.49
CA2 P00918 2/20 0.49
CA9 Q16790 2/20 0.49
TBXAS1 P24557 2/20 0.49
CYP11B1 P15538 1/20 0.49
CYP11B2 P19099 1/20 0.49
PORCN Q9H237 1/20 0.48
HTR2A P28223 1/20 0.48

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3990221 0.81 CYP3A4 (0.55) CYP3A4BAZ2BCYP2D6CYP2C9CYP1A2
SCHEMBL4757507 0.81 CYP3A4 (0.55) CYP3A4BAZ2BCYP2D6CYP2C9CYP1A2
SCHEMBL17315098 0.81 CYP3A4 (0.64) CYP3A4BAZ2BCYP2D6CYP2C9CYP1A2
SCHEMBL4661827 0.79 CYP3A4 (0.53) CYP3A4BAZ2BCYP2D6CYP2C9CYP1A2
SCHEMBL27814146 0.78 CYP3A4 (0.55) CYP3A4BAZ2BCYP2D6CYP2C9CYP1A2
SCHEMBL9451421 0.75 CYP2D6 (0.72) CYP3A4CYP2D6CYP2C9CYP1A2CYP2C19
SCHEMBL10512975 0.75 LMNA (0.62) CYP3A4BAZ2BCYP2D6CYP2C9CYP1A2
SCHEMBL5647102 0.74 ALDH1A1 (0.62) CYP3A4BAZ2BCYP2D6CYP2C9CYP1A2
SCHEMBL1931453 0.74 KMT2A (0.54) CYP19A1HTT
SCHEMBL2532397 0.74 LMNA (0.78) CYP3A4BAZ2BCYP2D6CYP2C9CYP1A2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-102127091-B Heterocyclic ring-containing schiff base compound TIANJIN INST PHARM RESEARCH 2012-11-21 CN disclosed
CN-102127091-A Heterocyclic ring-containing schiff base compound TIANJIN INST PHARM RESEARCH 2011-07-20 CN disclosed