SCHEMBL27835902

SCHEMBL27835902

CC(C)(O)C(CO)C(=N)C(=O)O

nearest known ligand 0.31

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
HMGCR P04035 1/20 0.31
CHRM1 P11229 1/20 0.31
TBXA2R P21731 1/20 0.31
ADRA1A P35348 1/20 0.31
ALDH1A1 P00352 1/20 0.31
TSHR P16473 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28390971 0.77 OR51E2 (0.38) HMGCRCHRM1TBXA2RADRA1AALDH1A1
SCHEMBL28146443 0.72 HMGCR (0.31) HMGCRCHRM1TBXA2RADRA1AALDH1A1
SCHEMBL27703766 0.65
SCHEMBL27653300 0.65 ALDH1A1 (0.39) ALDH1A1
SCHEMBL667279 0.64 OR51E2 (0.39) HMGCRCHRM1TBXA2RADRA1AALDH1A1
SCHEMBL13316605 0.64 OR51E2 (0.39) HMGCRCHRM1TBXA2RADRA1AALDH1A1
SCHEMBL27559021 0.64 CA2 (0.37) CHRM1ADRA1ATSHR
SCHEMBL27605345 0.64 CA2 (0.37) CHRM1ADRA1ATSHR
SCHEMBL27671851 0.64 CA2 (0.37) CHRM1ADRA1ATSHR
SCHEMBL16637322 0.62

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-102026974-B Tetrahydrocyclopenta[b]indole androgen receptor modulators LILLY CO ELI 2013-08-28 CN disclosed
CN-102026974-A Tetrahydrocyclopenta[b]indole androgen receptor modulators LILLY CO ELI 2011-04-20 CN disclosed