SCHEMBL27853045

SCHEMBL27853045

CC(=O)OC1CCNC(Cc2ccc(OC(F)(F)F)cc2)C1

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HTR2C P28335 2/20 0.44
CYP2D6 P10635 3/20 0.38
SMN1; SMN2 Q16637 3/20 0.38
LMNA P02545 1/20 0.38
MAPK1 P28482 1/20 0.38
HIF1A Q16665 1/20 0.38
MEN1 O00255 1/20 0.38
ALDH1A1 P00352 1/20 0.38
CYP2C9 P11712 1/20 0.38
CYP2C19 P33261 1/20 0.38
KMT2A Q03164 1/20 0.38
SLC2A1 P11166 1/20 0.38
EPHX2 P34913 4/20 0.37
HRH3 Q9Y5N1 2/20 0.37
EPHX1 P07099 1/20 0.37
FAAH O00519 2/20 0.36
TSHR P16473 1/20 0.36
CCNA2 P20248 1/20 0.36
CDK2 P24941 1/20 0.36
CCNA1 P78396 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL27852982 0.86 PPARG (0.38) CYP2D6SMN1; SMN2LMNAMAPK1HIF1A
SCHEMBL27853024 0.84 PLG (0.47) CYP2D6SMN1; SMN2LMNAMAPK1HIF1A
SCHEMBL27965419 0.82 CYP2D6 (0.37) CYP2D6SMN1; SMN2LMNAMAPK1HIF1A
SCHEMBL27869764 0.80 CYP2D6 (0.38) CYP2D6SMN1; SMN2LMNAMAPK1HIF1A
SCHEMBL581932 0.80 HTR2C (0.49) HTR2CSMN1; SMN2ALDH1A1EPHX2EPHX1
SCHEMBL27853003 0.79 KCNN4 (0.36) EPHX2
SCHEMBL27965683 0.79 ALDH1A1 (0.39) HTR2CCYP2D6SMN1; SMN2LMNAMAPK1
SCHEMBL27853046 0.78 HTR2C (0.45) HTR2CALDH1A1
SCHEMBL28794681 0.78 SMN1; SMN2 (0.41) SMN1; SMN2LMNAALDH1A1
Acetic Acid SCHEMBL27852948 0.78 POLB (0.52) HTR2CCYP2D6SMN1; SMN2LMNACYP2C9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-102459246-B Isoxazol-3 (2H) -one analogs as therapeutic agents ASTRAZENECA AB 2014-05-07 CN disclosed
CN-102459246-A Isoxazol-3 (2H) -one analogs as therapeutic agents ASTRAZENECA AB 2012-05-16 CN disclosed