SCHEMBL27869764

SCHEMBL27869764

CC(=O)OC1CCNC(Cc2ccc(C[SH](=O)=O)cc2)C1

nearest known ligand 0.38

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
CYP2D6 P10635 3/20 0.38
SMN1; SMN2 Q16637 3/20 0.38
LMNA P02545 1/20 0.38
MAPK1 P28482 1/20 0.38
HIF1A Q16665 1/20 0.38
MEN1 O00255 1/20 0.38
ALDH1A1 P00352 1/20 0.38
CYP2C9 P11712 1/20 0.38
CYP2C19 P33261 1/20 0.38
KMT2A Q03164 1/20 0.38
SLC2A1 P11166 1/20 0.38
PLG P00747 3/20 0.34
BACE1 P56817 1/20 0.33
POLB P06746 1/20 0.31
SLC6A2 P23975 1/20 0.31
SLC6A4 P31645 1/20 0.31
CCR3 P51677 1/20 0.31
SLC6A3 Q01959 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL27853024 0.85 PLG (0.47) CYP2D6SMN1; SMN2LMNAMAPK1HIF1A
SCHEMBL27965419 0.85 CYP2D6 (0.37) CYP2D6SMN1; SMN2LMNAMAPK1HIF1A
SCHEMBL27852982 0.82 PPARG (0.38) CYP2D6SMN1; SMN2LMNAMAPK1HIF1A
Hydrochloric Acid SCHEMBL27869800 0.82 CYP2D6 (0.33) CYP2D6SMN1; SMN2LMNAMAPK1HIF1A
SCHEMBL27853045 0.80 HTR2C (0.44) CYP2D6SMN1; SMN2LMNAMAPK1HIF1A
SCHEMBL27965683 0.80 ALDH1A1 (0.39) CYP2D6SMN1; SMN2LMNAMAPK1HIF1A
SCHEMBL27965650 0.78 BACE1 (0.47) PLGBACE1SLC6A2SLC6A4CCR3
SCHEMBL27853048 0.76 PLG (0.52) KMT2APLGBACE1SLC6A2SLC6A4
Hydrochloric Acid SCHEMBL27965754 0.76 BACE1 (0.38) CYP2D6SMN1; SMN2LMNAMAPK1HIF1A
SCHEMBL27869771 0.76 BACE1 (0.35) LMNAPLGBACE1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-102459246-B Isoxazol-3 (2H) -one analogs as therapeutic agents ASTRAZENECA AB 2014-05-07 CN disclosed
CN-102459246-A Isoxazol-3 (2H) -one analogs as therapeutic agents ASTRAZENECA AB 2012-05-16 CN disclosed