SCHEMBL2785997

SCHEMBL2785997

CC1(NC(=O)c2cncnc2)CC(O)C1

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
BDKRB1 P46663 4/20 0.39
TSHR P16473 1/20 0.38
KDM4E B2RXH2 3/20 0.38
HSD17B10 Q99714 1/20 0.38
HCAR2 Q8TDS4 1/20 0.37
VNN1 O95497 2/20 0.36
LATS1 O95835 1/20 0.35
LATS2 Q9NRM7 1/20 0.35
HDAC3 O15379 2/20 0.33
HDAC1 Q13547 2/20 0.33
HDAC2 Q92769 2/20 0.33
HDAC6 Q9UBN7 2/20 0.33
ABL1 P00519 1/20 0.33
BCAT2 O15382 1/20 0.33
BACE1 P56817 1/20 0.32
SIRT2 Q8IXJ6 1/20 0.32
HDAC4 P56524 1/20 0.32
HDAC7 Q8WUI4 1/20 0.32
HDAC10 Q969S8 1/20 0.32
HDAC11 Q96DB2 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL186482 0.83 BDKRB1 (0.42) BDKRB1TSHRKDM4EHSD17B10HCAR2
SCHEMBL2786986 0.80 BDKRB1 (0.38) BDKRB1TSHRKDM4EHSD17B10HCAR2
SCHEMBL185748 0.75 VNN1 (0.41) BDKRB1HCAR2VNN1ABL1BACE1
SCHEMBL20069112 0.75 BDKRB1 (0.38) BDKRB1HCAR2VNN1HDAC3HDAC1
SCHEMBL2787773 0.75 VNN1 (0.41) BDKRB1HCAR2VNN1ABL1BACE1
SCHEMBL20205895 0.72 BDKRB1 (0.36) BDKRB1HCAR2VNN1HDAC3HDAC1
SCHEMBL20147619 0.72 BDKRB1 (0.41) BDKRB1HCAR2VNN1HDAC3HDAC1
SCHEMBL20158441 0.70 BDKRB1 (0.39) BDKRB1VNN1HDAC3HDAC1HDAC2
SCHEMBL27363077 0.69 HCAR2 (0.38) BDKRB1KDM4EHCAR2ABL1BCAT2
SCHEMBL185415 0.68 BDKRB1 (0.47) BDKRB1TSHRKDM4EHSD17B10HCAR2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2010097374-A1 COMPOUNDS FOR USE AS BRADYKININ B1 ANTAGONISTS BOEHRINGER INGELHEIM INTERNATIONAL GMBH (DE) 2010-09-02 WO disclosed