SCHEMBL2786358

SCHEMBL2786358

COc1ccc(Oc2ccc(CNC(=O)C3(NC(=O)Oc4cncnc4)CCC(O)C3)cc2)c(C(F)(F)F)c1

nearest known ligand 0.39

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
P2RX7 Q99572 1/20 0.39
EPHX2 P34913 6/20 0.35
BDKRB1 P46663 2/20 0.35
POLB P06746 1/20 0.35
CCR2 P41597 3/20 0.34
ALDH1A1 P00352 1/20 0.34
L3MBTL1 Q9Y468 1/20 0.34
FAAH O00519 1/20 0.34
TRPV1 Q8NER1 1/20 0.34
PTPN7 P35236 2/20 0.33
DUSP3 P51452 2/20 0.33
KCNH2 Q12809 2/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2808220 0.95 P2RX7 (0.40) P2RX7EPHX2BDKRB1POLBCCR2
SCHEMBL2808204 0.94 P2RX7 (0.39) P2RX7EPHX2BDKRB1POLBALDH1A1
SCHEMBL2809672 0.93 P2RX7 (0.37) P2RX7EPHX2BDKRB1POLBCCR2
SCHEMBL13165653 0.92 BDKRB1 (0.44) P2RX7EPHX2BDKRB1POLB
SCHEMBL2810276 0.91 P2RX7 (0.38) P2RX7EPHX2BDKRB1POLBALDH1A1
SCHEMBL2812285 0.89 POLB (0.36) P2RX7EPHX2BDKRB1POLBALDH1A1
SCHEMBL2788425 0.88 EPHX2 (0.41) P2RX7EPHX2BDKRB1POLBALDH1A1
SCHEMBL2788200 0.87 BDKRB1 (0.38) P2RX7EPHX2BDKRB1POLBALDH1A1
SCHEMBL13165610 0.87 BDKRB1 (0.47) P2RX7EPHX2BDKRB1POLB
SCHEMBL2812521 0.87 BDKRB1 (0.38) P2RX7EPHX2BDKRB1POLBALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2010097374-A1 COMPOUNDS FOR USE AS BRADYKININ B1 ANTAGONISTS BOEHRINGER INGELHEIM INTERNATIONAL GMBH (DE) 2010-09-02 WO disclosed