SCHEMBL2787004

SCHEMBL2787004

CN[C@H]1CCc2cc(Br)ccc2C1

nearest known ligand 0.45

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
DRD2 P14416 1/20 0.45
DRD4 P21917 1/20 0.45
DRD3 P35462 1/20 0.45
CYP2C8 P10632 2/20 0.45
CYP2C9 P11712 2/20 0.45
KCNH2 Q12809 2/20 0.45
CYP2B6 P20813 1/20 0.45
ADRA2A P08913 4/20 0.44
PNMT P11086 4/20 0.44
ADRA2B P18089 3/20 0.44
ADRA2C P18825 3/20 0.44
HTR1D P28221 1/20 0.43
HTR1B P28222 1/20 0.43
CA1 P00915 4/20 0.41
CA2 P00918 4/20 0.41
ACHE P22303 4/20 0.41
HDAC8 Q9BY41 1/20 0.41
CYP11B2 P19099 1/20 0.40
CYP2D6 P10635 1/20 0.40
ASIC3 Q9UHC3 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL23306037 1.00 DRD2 (0.45) DRD2DRD4DRD3CYP2C8CYP2C9
SCHEMBL2876799 0.85 PNMT (0.49) ADRA2APNMTADRA2BADRA2C
SCHEMBL13950761 0.83 CYP2C8 (0.42) CYP2C8CYP2C9KCNH2CYP2B6ADRA2A
SCHEMBL29113500 0.82 DRD2 (0.48) DRD2DRD3CYP2C8CYP2C9KCNH2
SCHEMBL20909682 0.81 DRD2 (0.46) DRD2DRD4DRD3HTR1DHTR1B
SCHEMBL12778356 0.80 CYP2C8 (0.41) CYP2C8CYP2C9KCNH2CYP2B6ADRA2A
SCHEMBL2086346 0.80 CYP2C8 (0.41) CYP2C8CYP2C9KCNH2CYP2B6ADRA2A
SCHEMBL6839556 0.79 CA1 (0.62) DRD2DRD4DRD3HTR1DHTR1B
SCHEMBL20722746 0.78 CA1 (0.50) CYP2C8CYP2C9KCNH2CYP2B6ADRA2A
SCHEMBL20722885 0.78 CA1 (0.50) CYP2C8CYP2C9KCNH2CYP2B6ADRA2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2396300-A1 NEW SUBSTITUTED TETRAHYDRONAPTHALENES, METHOD FOR THE PRODUCTION THEREOF, AND USE THEREOF AS DRUGS SANOFI (FR) 2011-12-21 EP disclosed
WO-2010092153-A1 NEW SUBSTITUTED TETRAHYDRONAPTHALENES, METHOD FOR THE PRODUCTION THEREOF, AND USE THEREOF AS DRUGS SANOFI-AVENTIS (FR) 2010-08-19 WO disclosed