SCHEMBL27872202

SCHEMBL27872202

O=[N+]([O-])c1ccc(-c2cc(CCBr)on2)cc1

nearest known ligand 0.50

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CA12 O43570 2/20 0.50
CA9 Q16790 2/20 0.50
SIRT2 Q8IXJ6 1/20 0.50
CXCR1 P25024 1/20 0.47
DRD2 P14416 4/20 0.42
DRD4 P21917 4/20 0.42
DRD3 P35462 4/20 0.42
MAPT P10636 5/20 0.42
NPC1 O15118 3/20 0.42
RAB9A P51151 3/20 0.42
NOTUM Q6P988 4/20 0.40
CYP1A2 P05177 1/20 0.39
CYP3A4 P08684 1/20 0.39
CYP2D6 P10635 1/20 0.39
CYP2C9 P11712 1/20 0.39
CYP2C19 P33261 1/20 0.39
HTT P42858 1/20 0.39
CHRNB2 P17787 1/20 0.39
CHRNA5 P30532 1/20 0.39
CHRNA4 P43681 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL17978447 0.83 CA12 (0.48) CA12CA9SIRT2CXCR1DRD2
SCHEMBL1220104 0.82 CA12 (0.52) CA12CA9SIRT2CXCR1MAPT
SCHEMBL2920882 0.82 NOTUM (0.60) CA12CA9SIRT2CXCR1MAPT
SCHEMBL189588 0.82 NOTUM (0.60) CA12CA9SIRT2CXCR1MAPT
SCHEMBL19403807 0.79 CXCR1 (0.50) CA12CA9SIRT2CXCR1MAPT
SCHEMBL27789238 0.77 NOTUM (0.66) SIRT2MAPTNPC1RAB9ANOTUM
SCHEMBL23881879 0.77 NOTUM (0.64) DRD2DRD4DRD3MAPTNPC1
SCHEMBL3822977 0.75 GSK3B (0.51) CA12CA9SIRT2CXCR1MAPT
SCHEMBL16549592 0.74 RAB9A (0.54) CA12CA9CXCR1MAPTNPC1
SCHEMBL3459689 0.74 CXCR1 (0.49) CA12CA9CXCR1MAPTNPC1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-102690241-B Benzoyl urea compound containing isoxazoline and isoxazole structure, and preparation and application thereof UNIV NANKAI 2014-07-09 CN disclosed
CN-102690241-A Benzoyl urea compound containing isoxazoline and isoxazole structure, and preparation and application thereof UNIV NANKAI 2012-09-26 CN disclosed