SCHEMBL2787488

SCHEMBL2787488

NC1(OC(=O)O)CC(OCc2ccccc2)C1

nearest known ligand 0.45

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
GRM2 Q14416 1/20 0.45
GRM3 Q14832 1/20 0.45
DPP4 P27487 1/20 0.43
EPHX2 P34913 2/20 0.43
CTSL P07711 1/20 0.41
CTSB P07858 1/20 0.41
CTSK P43235 1/20 0.41
ALDH1A1 P00352 2/20 0.41
OPRM1 P35372 2/20 0.40
OPRL1 P41146 2/20 0.40
SLC1A3 P43003 2/20 0.39
SLC1A2 P43004 2/20 0.39
SLC1A1 P43005 2/20 0.39
MEN1 O00255 1/20 0.39
CYP1A2 P05177 1/20 0.39
CYP2D6 P10635 1/20 0.39
CYP2C9 P11712 1/20 0.39
CYP2C19 P33261 1/20 0.39
KMT2A Q03164 1/20 0.39
PDPK1 O15530 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL27917553 0.86 OPRM1 (0.41) GRM2GRM3DPP4EPHX2CTSL
SCHEMBL14409083 0.81 GRM2 (0.47) GRM2GRM3DPP4EPHX2CTSL
SCHEMBL296907 0.81 GRM2 (0.47) GRM2GRM3DPP4EPHX2CTSL
SCHEMBL22509327 0.81 EPHX2 (0.43) GRM2GRM3DPP4EPHX2CTSL
SCHEMBL15316801 0.80 DPP4 (0.44) GRM2GRM3DPP4EPHX2CTSL
SCHEMBL28055036 0.80 DPP4 (0.50) GRM2GRM3DPP4EPHX2CTSL
SCHEMBL7936878 0.78 DPP4 (0.46) GRM2GRM3DPP4EPHX2CTSL
SCHEMBL2640274 0.78 EPHX2 (0.47) GRM2GRM3DPP4EPHX2CTSL
SCHEMBL31471412 0.77 DPP4 (0.44) GRM2GRM3DPP4EPHX2CTSL
SCHEMBL23274871 0.77 EPHX2 (0.44) GRM2GRM3DPP4EPHX2CTSL

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2010097374-A1 COMPOUNDS FOR USE AS BRADYKININ B1 ANTAGONISTS BOEHRINGER INGELHEIM INTERNATIONAL GMBH (DE) 2010-09-02 WO disclosed