SCHEMBL27883271

SCHEMBL27883271

Cc1cccc(C=O)c1-n1ccnn1

nearest known ligand 0.43

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 1/20 0.43
TSHR P16473 1/20 0.43
NOTUM Q6P988 9/20 0.41
HCRTR1 O43613 4/20 0.41
HCRTR2 O43614 4/20 0.41
KEAP1 Q14145 1/20 0.37
TRIM24 O15164 1/20 0.34
TRIM33 Q9UPN9 1/20 0.34
MEN1 O00255 1/20 0.32
LMNA P02545 1/20 0.32
THRB P10828 1/20 0.32
BLM P54132 1/20 0.32
KMT2A Q03164 1/20 0.32
TDP1 Q9NUW8 1/20 0.32
MAP3K5 Q99683 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28858824 0.83 NOTUM (0.49) ALDH1A1NOTUMKEAP1MEN1KMT2A
SCHEMBL18367778 0.78 NOTUM (0.41) ALDH1A1TSHRNOTUMHCRTR1HCRTR2
SCHEMBL3388189 0.76 NOTUM (0.47) NOTUMHCRTR1HCRTR2KEAP1
SCHEMBL6428991 0.76 NOTUM (0.44) TSHRNOTUMHCRTR1HCRTR2KEAP1
SCHEMBL27883266 0.75 HCRTR1 (0.54) ALDH1A1NOTUMHCRTR1HCRTR2KEAP1
SCHEMBL1586907 0.74 HCRTR1 (0.53) ALDH1A1NOTUMHCRTR1HCRTR2MEN1
SCHEMBL14939847 0.73 ALDH1A1 (0.48) ALDH1A1TSHRHCRTR1HCRTR2TRIM24
SCHEMBL2854803 0.73 NOTUM (0.42) ALDH1A1TSHRNOTUMHCRTR1HCRTR2
SCHEMBL17910085 0.73 HCRTR1 (0.52) NOTUMHCRTR1HCRTR2KEAP1TDP1
SCHEMBL1586174 0.72 TSHR (0.43) ALDH1A1TSHRNOTUMHCRTR1HCRTR2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-102781942-B Octahydro pyrrolo-[3,4-c] pyrroles is replaced as two of orexin receptor modulators JANSSEN PHARMACEUTICA N.V. (BE) 2015-09-23 CN claimed
CN-102781942-A Disubstituted octahy-dropyrrolo [3,4-c]pyrroles as orexin receptor modulators JANSSEN PHARMACEUTICA NV 2012-11-14 CN claimed
CN-102781942-B Octahydro pyrrolo-[3,4-c] pyrroles is replaced as two of orexin receptor modulators JANSSEN PHARMACEUTICA N.V. (BE) 2015-09-23 CN disclosed
CN-102781942-A Disubstituted octahy-dropyrrolo [3,4-c]pyrroles as orexin receptor modulators JANSSEN PHARMACEUTICA NV 2012-11-14 CN disclosed