SCHEMBL27883282

SCHEMBL27883282

O=C(c1cc(F)ccc1I)c1cc(F)ccc1I

nearest known ligand 0.50

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
CES2 O00748 7/20 0.50
CES1 P23141 7/20 0.50
KEAP1 Q14145 1/20 0.45
TTR P02766 1/20 0.40
ANO1 Q5XXA6 1/20 0.38
ALDH1A1 P00352 1/20 0.38
HTT P42858 1/20 0.38
HPGD P15428 1/20 0.36
MAOB P27338 1/20 0.35
CA3 P07451 1/20 0.34
CA6 P23280 1/20 0.34
CA5A P35218 1/20 0.34
CA9 Q16790 1/20 0.34
CA14 Q9ULX7 1/20 0.34
CA5B Q9Y2D0 1/20 0.34
HDAC1 Q13547 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1150930 0.84 KEAP1 (0.59) CES2CES1KEAP1TTRANO1
SCHEMBL30762574 0.84 KEAP1 (0.59) CES2CES1KEAP1TTRANO1
SCHEMBL28423060 0.83 CES2 (0.47) CES2CES1KEAP1TTRANO1
SCHEMBL1804347 0.83 KEAP1 (0.47) CES2CES1KEAP1TTRANO1
SCHEMBL2584947 0.83 CES2 (0.47) CES2CES1KEAP1TTRANO1
SCHEMBL31448305 0.83 CES2 (0.47) CES2CES1KEAP1TTRANO1
SCHEMBL27883251 0.82 CES2 (0.50) CES2CES1KEAP1TTRALDH1A1
SCHEMBL15273748 0.79 CES2 (0.44) CES2CES1KEAP1TTRANO1
SCHEMBL31274973 0.78 CES2 (0.42) CES2CES1KEAP1TTRALDH1A1
SCHEMBL1151008 0.78 SLC6A4 (0.47) CES2CES1ALDH1A1HTTHPGD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-102781942-A Disubstituted octahy-dropyrrolo [3,4-c]pyrroles as orexin receptor modulators JANSSEN PHARMACEUTICA NV 2012-11-14 CN disclosed