SCHEMBL2789018

SCHEMBL2789018

COC[C@](C)(NC(=O)c1cncnc1)C(=O)O

nearest known ligand 0.38

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HCAR2 Q8TDS4 1/20 0.38
BCAT2 O15382 1/20 0.33
CTSL P07711 1/20 0.33
POLB P06746 1/20 0.33
ITGAV P06756 1/20 0.32
NPSR1 Q6W5P4 1/20 0.32
GPR132 Q9UNW8 1/20 0.32
ACACB O00763 1/20 0.32
MAPK1 P28482 1/20 0.32
SMN1; SMN2 Q16637 1/20 0.32
CYP1A2 P05177 1/20 0.32
CYP3A4 P08684 1/20 0.32
CYP2C19 P33261 1/20 0.32
HCAR3 P49019 1/20 0.31
ATM Q13315 1/20 0.31
ALDH1A1 P00352 1/20 0.31
HPGDS O60760 1/20 0.31
MEN1 O00255 1/20 0.31
KMT2A Q03164 1/20 0.31
PRSS1 P07477 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2787762 1.00 HCAR2 (0.38) HCAR2BCAT2CTSLPOLBITGAV
SCHEMBL2787521 1.00 HCAR2 (0.38) HCAR2BCAT2CTSLPOLBITGAV
SCHEMBL2790368 0.87 HCAR2 (0.37) HCAR2BCAT2CTSLPOLBITGAV
SCHEMBL2789685 0.77 HCAR2 (0.36) HCAR2BCAT2CTSLPOLBITGAV
SCHEMBL14865358 0.76 HCAR2 (0.47) HCAR2BCAT2CTSLPOLBITGAV
SCHEMBL2788519 0.74 MAPK1 (0.43) ACACBMAPK1SMN1; SMN2CYP1A2CYP3A4
SCHEMBL2787725 0.72 MAPK1 (0.33) HCAR2MAPK1SMN1; SMN2ALDH1A1
SCHEMBL19877014 0.71 NPC1 (0.46) HCAR2POLBATM
SCHEMBL9010820 0.70 SMN1; SMN2 (0.33) HCAR2CTSLITGAVNPSR1ACACB
SCHEMBL5768937 0.69 KMT2A (0.42) HCAR2CTSLPOLBITGAVCYP1A2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2010097374-A1 COMPOUNDS FOR USE AS BRADYKININ B1 ANTAGONISTS BOEHRINGER INGELHEIM INTERNATIONAL GMBH (DE) 2010-09-02 WO disclosed