SCHEMBL9010820

SCHEMBL9010820

CCC(C)(NC(=O)c1cncnc1)C(=O)C(Br)Br

nearest known ligand 0.35

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SMN1; SMN2 Q16637 3/20 0.33
HTT P42858 3/20 0.33
MAPT P10636 2/20 0.33
MAPK1 P28482 2/20 0.33
BDKRB1 P46663 1/20 0.33
ACACB O00763 1/20 0.33
CNR2 P34972 1/20 0.33
NPC1 O15118 1/20 0.33
TSHR P16473 1/20 0.33
RAB9A P51151 1/20 0.33
CYP1A2 P05177 1/20 0.33
CYP3A4 P08684 1/20 0.33
CYP2C19 P33261 1/20 0.33
HCAR2 Q8TDS4 1/20 0.33
CTSL P07711 1/20 0.33
KDM4E B2RXH2 1/20 0.33
ITGAV P06756 1/20 0.32
GFER P55789 1/20 0.32
NPSR1 Q6W5P4 1/20 0.32
HDAC3 O15379 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9010890 0.78 ERAP1 (0.34) HTTCNR2CYP2C19
SCHEMBL8156479 0.77 GRN (0.45) RAB9A
SCHEMBL8167643 0.75 ALDH1A1 (0.33) HTTMAPTNPC1CYP1A2CYP3A4
SCHEMBL8060065 0.74 HSD11B1 (0.36) HTTMAPTTSHRCYP1A2CYP3A4
SCHEMBL19877014 0.70 NPC1 (0.46) CNR2NPC1RAB9AHCAR2
SCHEMBL2787762 0.70 HCAR2 (0.38) SMN1; SMN2MAPK1ACACBCYP1A2CYP3A4
SCHEMBL2789018 0.70 HCAR2 (0.38) SMN1; SMN2MAPK1ACACBCYP1A2CYP3A4
SCHEMBL2787521 0.70 HCAR2 (0.38) SMN1; SMN2MAPK1ACACBCYP1A2CYP3A4
SCHEMBL9010839 0.69 ALDH1A1 (0.36) SMN1; SMN2MAPTNPC1RAB9AKDM4E
SCHEMBL2790368 0.69 HCAR2 (0.37) SMN1; SMN2MAPK1ACACBCNR2HCAR2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 7 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5547984-A FUNGICIDES ROHM AND HAAS COMPANY (US) 1996-08-20 US disclosed
US-5529978-A FUNGICIDE ROHM AND HAAS COMPANY (US) 1996-06-25 US disclosed
US-5344978-A Fungicides ROHM AND HAAS COMPANY (US) 1994-09-06 US disclosed
US-5196046-A N-acetonyl-substituted-amides ROHM AND HAAS COMPANY (US) 1993-03-23 US disclosed
EP-0170498-B1 N-ACETONYL-SUBSTITUTED-AMIDES, COMPOSITIONS CONTAINING THEM AND THEIR USE IN COMBATING FUNGI ROHM AND HAAS COMPANY (US) 1991-09-11 EP disclosed
US-4863940-A N-acetonyl-substituted amides and phytopathogenic fungicidal use thereof ROHM AND HAAS (US) 1989-09-05 US disclosed
EP-0170498-A2 N-acetonyl-substituted-amides, compositions containing them and their use in combating fungi ROHM AND HAAS COMPANY (US) 1986-02-05 EP disclosed