SCHEMBL14865358

SCHEMBL14865358

CC(C)(NC(=O)c1cncnc1)C(=O)O

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HCAR2 Q8TDS4 1/20 0.47
EGLN1 Q9GZT9 1/20 0.41
EGLN3 Q9H6Z9 1/20 0.41
BCAT2 O15382 1/20 0.40
POLB P06746 1/20 0.39
KDM4E B2RXH2 2/20 0.37
MAPT P10636 1/20 0.36
CTSL P07711 1/20 0.35
KDM4C Q9H3R0 1/20 0.34
LATS1 O95835 1/20 0.34
ITGAV P06756 1/20 0.34
ALDH1A1 P00352 1/20 0.33
MRGPRX4 Q96LA9 1/20 0.33
BRAF P15056 1/20 0.33
LCK P06239 1/20 0.33
KIT P10721 1/20 0.33
SRC P12931 1/20 0.33
MAPK14 Q16539 1/20 0.33
HDAC3 O15379 1/20 0.33
HDAC1 Q13547 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL19877014 0.76 NPC1 (0.46) HCAR2POLB
SCHEMBL2787762 0.76 HCAR2 (0.38) HCAR2BCAT2POLBCTSLITGAV
SCHEMBL2787521 0.76 HCAR2 (0.38) HCAR2BCAT2POLBCTSLITGAV
SCHEMBL2789018 0.76 HCAR2 (0.38) HCAR2BCAT2POLBCTSLITGAV
SCHEMBL2790368 0.75 HCAR2 (0.37) HCAR2EGLN1BCAT2POLBCTSL
SCHEMBL2871262 0.75 HCAR2 (0.46) HCAR2BCAT2KDM4EBRAFLCK
SCHEMBL343830 0.75 POLB (0.65) POLBKDM4EMRGPRX4HDAC3HDAC1
SCHEMBL2789685 0.74 HCAR2 (0.36) HCAR2BCAT2POLBCTSLITGAV
SCHEMBL2787729 0.73 HCAR2 (0.35) HCAR2BCAT2POLBCTSLITGAV
Trifluoroacetic Acid SCHEMBL29699595 0.73 HCAR2 (0.50) HCAR2BCAT2KDM4ECTSLALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2401256-B1 Compounds as bradykinin B1 antagonists BOEHRINGER INGELHEIM INT (DE) 2013-04-17 EP disclosed