SCHEMBL27900552

SCHEMBL27900552

O=CN(c1ncc(-c2ccc(NC(=O)c3cscn3)cc2)s1)N1CCC(=Cc2ccccn2)CC1

nearest known ligand 0.37

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
GRM4 Q14833 2/20 0.37
NAMPT P43490 1/20 0.36
NPC1 O15118 5/20 0.34
RAB9A P51151 5/20 0.34
SMN1; SMN2 Q16637 3/20 0.34
MAPT P10636 1/20 0.34
PKM P14618 1/20 0.34
HTT P42858 1/20 0.34
KLF5 Q13887 1/20 0.34
PIM1 P11309 1/20 0.34
GRM1 Q13255 1/20 0.34
PTGDR2 Q9Y5Y4 1/20 0.33
HPGD P15428 2/20 0.33
MEN1 O00255 1/20 0.33
KMT2A Q03164 1/20 0.33
TP53 P04637 1/20 0.33
MAPK1 P28482 1/20 0.33
ROCK2 O75116 1/20 0.32
ROCK1 Q13464 1/20 0.32
KDR P35968 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL460271 0.82 NAMPT (0.44) GRM4NAMPTNPC1RAB9ASMN1; SMN2
SCHEMBL27900550 0.81 CSNK2A1 (0.38)
SCHEMBL28802184 0.74 KDM4E (0.33) NPC1RAB9ASMN1; SMN2MAPTPKM
SCHEMBL27918356 0.72 OGA (0.34) NPC1RAB9AMAPTKMT2AMAPK1
SCHEMBL27918264 0.69 SRD5A2 (0.35) HPGDKDM4EALDH1A1
SCHEMBL28802187 0.69 GRM4 (0.37) GRM4NAMPTNPC1RAB9ASMN1; SMN2
SCHEMBL15070397 0.68 GRM4 (0.47) GRM4NPC1RAB9ASMN1; SMN2MAPT
SCHEMBL459963 0.66 CNR2 (0.49) NAMPTKDRFLT3
SCHEMBL28802159 0.65 LDHA (0.39) NPC1RAB9ASMN1; SMN2TP53
SCHEMBL28802153 0.65 GRM4 (0.46) GRM4NPC1RAB9ASMN1; SMN2MAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-103080086-B Prostaglandin D synthase inhibitory piperidine compounds TAIHO PHARMACEUTICAL CO LTD 2014-11-05 CN claimed
CN-103080086-B Prostaglandin D synthase inhibitory piperidine compounds TAIHO PHARMACEUTICAL CO LTD 2014-11-05 CN disclosed
CN-103080086-A Prostaglandin D synthase inhibitory piperidine compounds TAIHO PHARMACEUTICAL CO LTD 2013-05-01 CN disclosed