SCHEMBL27902017

SCHEMBL27902017

O=C(O)CN(Cc1cc(C(F)(F)F)cc(C(F)(F)F)c1)Cc1cc2ccccc2nc1Cl

nearest known ligand 0.41

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
TACR1 P25103 12/20 0.41
KMT2A Q03164 2/20 0.41
L3MBTL1 Q9Y468 1/20 0.41
GPBAR1 Q8TDU6 4/20 0.39
MEN1 O00255 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5624217 0.86 TACR1 (0.38) TACR1KMT2AGPBAR1
SCHEMBL28034153 0.81 TACR1 (0.43) TACR1GPBAR1
SCHEMBL5666117 0.80 MAPT (0.38) TACR1L3MBTL1GPBAR1
SCHEMBL14602919 0.78 CETP (0.46) TACR1GPBAR1
SCHEMBL13673129 0.77 TACR1 (0.48) TACR1KMT2AL3MBTL1MEN1
SCHEMBL7959904 0.76 TACR1 (0.49) TACR1KMT2AL3MBTL1MEN1
SCHEMBL15706233 0.73 CETP (0.41) TACR1KMT2AGPBAR1
SCHEMBL5802941 0.72 TACR1 (0.52) TACR1KMT2AL3MBTL1GPBAR1
SCHEMBL9408665 0.72 TDP1 (0.47) TACR1KMT2AL3MBTL1MEN1
SCHEMBL9408639 0.72 TDP1 (0.47) TACR1KMT2AL3MBTL1MEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-103102303-B As the benzyl amine derivative of CETP inhibitor DR. REDDY'S LABORATORIES LTD. (IN) 2015-10-28 CN disclosed
CN-103102303-A Benzylamine derivatives as CETP inhibitors REDDY US THERAPEUTICS INC 2013-05-15 CN disclosed