SCHEMBL27903451

SCHEMBL27903451

NC(=O)c1cccc(C2CC2)c1N1CCN(C2CCC2)CC1

nearest known ligand 0.52

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
PARP1 P09874 15/20 0.52
CYP2D6 P10635 1/20 0.48
CYP2B6 P20813 1/20 0.48
PARP2 Q9UGN5 4/20 0.44
KDM2B Q8NHM5 3/20 0.41
HRH3 Q9Y5N1 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL12490895 0.85 NPC1 (0.53) PARP1CYP2D6CYP2B6PARP2
SCHEMBL27903450 0.74 PARP1 (0.51) PARP1CYP2D6CYP2B6PARP2HRH3
SCHEMBL30839562 0.74 PARP1 (0.50) PARP1CYP2D6CYP2B6PARP2
SCHEMBL13806171 0.71 AURKA (0.44) PARP1PARP2
SCHEMBL30666294 0.71 KDM4E (0.39) PARP1PARP2
SCHEMBL3682185 0.70 NPC1 (0.62) PARP1PARP2
Hydrochloric Acid SCHEMBL4253332 0.70 AURKA (0.44) PARP1PARP2
SCHEMBL16372150 0.70 PARP2 (0.47) PARP1CYP2D6CYP2B6PARP2KDM2B
SCHEMBL13816304 0.69 AURKA (0.43) PARP1PARP2
SCHEMBL4554366 0.69 KDM2B (0.43) PARP1KDM2BHRH3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-103168027-A Process for preparing cyclopropyl amide derivatives and intermediates related thereto ASTRAZENECA AB 2013-06-19 CN disclosed
CN-102869651-A New crystalline form of a cyclopropyl benzamide derivative ASTRAZENECA AB 2013-01-09 CN disclosed