SCHEMBL2790767

SCHEMBL2790767

COCCCn1c([C@@H]2CCCN(C(=O)C[C@@H](Cc3ccc(-c4ccc(NCCO)nc4)cc3)NC(=O)O)C2)c(C)c2cccc(F)c21

nearest known ligand 0.31

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
MAPK1 P28482 2/20 0.31
ITGB1 P05556 1/20 0.31
ITGA4 P13612 1/20 0.31
ADRA1A P35348 2/20 0.31
PROKR1 Q8TCW9 1/20 0.31
ITGB3 P05106 1/20 0.31
ITGAV P06756 1/20 0.31
DRD2 P14416 1/20 0.30
DRD3 P35462 1/20 0.30
MMEL1 Q495T6 1/20 0.30
BTK Q06187 1/20 0.30
PDPK1 O15530 1/20 0.30
BDKRB1 P46663 2/20 0.30
ALDH1A1 P00352 1/20 0.30
TSHR P16473 1/20 0.30
KMT2A Q03164 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2789843 1.00 MAPK1 (0.31) MAPK1ITGB1ITGA4ADRA1APROKR1
SCHEMBL7900800 0.93 ALOX5AP (0.30)
SCHEMBL7898811 0.93 ALOX5AP (0.30)
SCHEMBL2789049 0.92 DPP4 (0.34) MAPK1ITGB1ITGA4ADRA1APROKR1
SCHEMBL2789767 0.92 DPP4 (0.34) MAPK1ITGB1ITGA4ADRA1APROKR1
SCHEMBL2791634 0.92 DPP4 (0.34) MAPK1ITGB1ITGA4ADRA1APROKR1
SCHEMBL2789770 0.92 DPP4 (0.34) MAPK1ITGB1ITGA4ADRA1APROKR1
SCHEMBL2791931 0.89 SCN9A (0.33) MAPK1ITGB1ITGA4PROKR1MMEL1
SCHEMBL2788040 0.85 BTK (0.33) MAPK1ITGB1ITGA4ADRA1APROKR1
SCHEMBL2791623 0.85 FPR2 (0.34) PROKR1ITGB3ALDH1A1TSHRKMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2010111634-A2 RENIN INHIBITORS TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2010-09-30 WO disclosed