SCHEMBL27908554

SCHEMBL27908554

O=[C]c1ccc(C(F)(F)F)cc1O

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MEN1 O00255 4/20 0.44
KMT2A Q03164 4/20 0.44
CES2 O00748 4/20 0.40
HSP90AA1 P07900 2/20 0.39
MAPT P10636 2/20 0.39
CYP1A2 P05177 1/20 0.39
CYP3A4 P08684 1/20 0.39
CYP2C9 P11712 1/20 0.39
TSHR P16473 1/20 0.39
NFKB1 P19838 1/20 0.39
CYP2C19 P33261 1/20 0.39
BLM P54132 1/20 0.39
PMP22 Q01453 1/20 0.39
KCNMA1 Q12791 1/20 0.39
NPSR1 Q6W5P4 1/20 0.39
KDM4E B2RXH2 2/20 0.38
HSD17B10 Q99714 2/20 0.38
ALDH1A1 P00352 1/20 0.38
HPGD P15428 1/20 0.38
NQO2 P16083 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2140819 0.78 PDE2A (0.42) MEN1KMT2ACES2KDM4EHSD17B10
SCHEMBL3033286 0.78 PDE2A (0.39) MEN1KMT2ACES2MAPTKDM4E
SCHEMBL2703782 0.78 CES2 (0.50) CES2AR
SCHEMBL3032872 0.76 MRGPRX4 (0.47) MEN1KMT2AMAPTTSHRALDH1A1
SCHEMBL13464023 0.74 ALDH1A1 (0.42) MEN1KMT2ACES2KDM4EALDH1A1
SCHEMBL483405 0.73 IDO1 (0.41) MEN1KMT2ACES2TSHRKDM4E
SCHEMBL6387748 0.73 CES2 (0.50) MEN1KMT2ACES2TSHRKDM4E
SCHEMBL187014 0.73 NQO2 (0.61) MEN1KMT2ACES2HSP90AA1MAPT
SCHEMBL14307167 0.72 MEN1 (0.44) MEN1KMT2ACES2HSP90AA1MAPT
SCHEMBL2515789 0.72 PTGDR2 (0.43) MEN1KMT2ACYP1A2CYP3A4TSHR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-103145662-A N-substituted animobutyrolactone derivatives and uses thereof SHENZHEN WANHE PHARMACEUTICAL CO LTD 2013-06-12 CN claimed
CN-103145662-B N-substituted animobutyrolactone derivatives and uses thereof SHENZHEN WANHE PHARMACEUTICAL CO LTD 2014-07-16 CN disclosed
CN-103145662-A N-substituted animobutyrolactone derivatives and uses thereof SHENZHEN WANHE PHARMACEUTICAL CO LTD 2013-06-12 CN disclosed