SCHEMBL27909660

SCHEMBL27909660

COc1ccc(CN2CC=C(c3c[nH]c4ccc(OC)cc34)CC2)cc1

nearest known ligand 1.00 ✓ in ChEMBL — recovers established targets

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
HTR1A P08908 17/20 1.00
DRD2 P14416 16/20 1.00
HTR2A P28223 5/20 0.72
SLC6A4 P31645 1/20 0.69
DRD1 P21728 1/20 0.66
DRD3 P35462 1/20 0.66
OPRM1 P35372 1/20 0.64
OPRK1 P41145 1/20 0.64
HTT P42858 1/20 0.60

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL27909555 0.94 HTR1A (0.88) HTR1ADRD2HTR2ASLC6A4DRD1
SCHEMBL4194997 0.94 HTR1A (1.00) HTR1ADRD2HTR2ASLC6A4DRD1
SCHEMBL27860653 0.92 HTR1A (0.85) HTR1ADRD2HTR2ASLC6A4DRD1
SCHEMBL4336592 0.90 HTR1A (0.82) HTR1ADRD2HTR2ASLC6A4DRD1
SCHEMBL13944275 0.90 HTR1A (0.80) HTR1ADRD2HTR2ASLC6A4DRD1
SCHEMBL11313868 0.86 HTR1A (0.75) HTR1ADRD2HTR2ASLC6A4DRD1
SCHEMBL11786344 0.85 HTR1A (0.85) HTR1ADRD2HTR2ADRD1DRD3
SCHEMBL7649906 0.82 HTR1A (0.83) HTR1ADRD2HTR2AOPRM1OPRK1
SCHEMBL7704740 0.82 SLC6A4 (1.00) HTR1ADRD2SLC6A4
SCHEMBL8553783 0.81 HTR1A (0.81) HTR1ADRD2HTR2ASLC6A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-102276581-B N-substituted tetrahydropyridine bound indole compound as well as preparation method and application thereof UNIV SHANGHAI 2013-06-12 CN disclosed