SCHEMBL7649906

SCHEMBL7649906

C1=C(c2c[nH]c3ccc(OCc4ccccc4)cc23)CCN(Cc2ccccc2)C1

nearest known ligand 0.83

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
HTR1A P08908 16/20 0.83
DRD2 P14416 15/20 0.83
HTR2A P28223 4/20 0.83
OPRM1 P35372 1/20 0.72
OPRK1 P41145 1/20 0.72
HTT P42858 1/20 0.69
ACHE P22303 1/20 0.60

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4194997 0.89 HTR1A (1.00) HTR1ADRD2HTR2AOPRM1OPRK1
SCHEMBL5365266 0.87 SLC6A4 (0.69) HTR1ADRD2HTR2A
SCHEMBL7536094 0.85 OPRM1 (0.78) HTR1ADRD2HTR2AOPRM1OPRK1
SCHEMBL14280720 0.84 OPRM1 (1.00) HTR1ADRD2HTR2AOPRM1OPRK1
SCHEMBL9527241 0.83 OPRM1 (0.78) HTR1ADRD2HTR2AOPRM1OPRK1
SCHEMBL6133368 0.83 DRD2 (0.71) HTR1ADRD2HTR2A
SCHEMBL16801500 0.82 HTR1A (0.61) HTR1ADRD2HTR2AOPRM1OPRK1
SCHEMBL7543848 0.82 HTR1A (1.00) HTR1ADRD2HTR2AOPRM1OPRK1
SCHEMBL27909660 0.82 HTR1A (1.00) HTR1ADRD2HTR2AOPRM1OPRK1
SCHEMBL7465475 0.81 HTR1A (0.57) HTR1ADRD2HTR2AOPRM1OPRK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6476028-B1 Compounds and methods SMITHKLINE BEECHAM CORPORATION 2002-11-05 US claimed
CN-102796075-B Benzocycloheptenes derivative as well as preparation method and medical application thereof INST PHARM & TOXICOLOGY AMMS 2014-03-12 CN disclosed
CN-101481323-B Benzocycloheptenes derivatives, preparation method and medical application thereof POISON MED INST PLA MED ACAD 2013-11-20 CN disclosed
CN-102796075-A Benzocycloheptenes derivative as well as preparation method and medical application thereof INST PHARM & TOXICOLOGY AMMS 2012-11-28 CN disclosed
US-6476028-B1 Compounds and methods SMITHKLINE BEECHAM CORPORATION 2002-11-05 US disclosed