SCHEMBL27913634

SCHEMBL27913634

Cc1onc(-c2ccc(F)cc2)c1C(=O)c1c(-c2ccc(F)cc2)noc1C

nearest known ligand 0.60

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
GPBAR1 Q8TDU6 2/20 0.60
LMNA P02545 2/20 0.55
KMT2A Q03164 4/20 0.54
GAA P10253 2/20 0.54
MEN1 O00255 2/20 0.54
TSHR P16473 1/20 0.52
KDM4E B2RXH2 2/20 0.52
ALDH1A1 P00352 1/20 0.52
PTGS2 P35354 2/20 0.51
BACE1 P56817 3/20 0.50
NPC1 O15118 1/20 0.47
ATM Q13315 1/20 0.47
GABRA5 P31644 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL457706 0.89 GPBAR1 (0.59) GPBAR1LMNAKMT2AGAAMEN1
SCHEMBL2475844 0.89 GPBAR1 (0.59) GPBAR1LMNAKMT2AGAAMEN1
Hydrochloric Acid SCHEMBL3981907 0.87 GPBAR1 (0.57) GPBAR1LMNAKMT2AGAAMEN1
SCHEMBL3068021 0.87 GPBAR1 (0.61) GPBAR1LMNAKMT2AGAAMEN1
SCHEMBL4718673 0.87 KMT2A (0.72) GPBAR1LMNAKMT2AGAAMEN1
Hydrochloric Acid SCHEMBL30684627 0.86 KMT2A (0.70) GPBAR1LMNAKMT2AGAAMEN1
SCHEMBL17736156 0.85 GPBAR1 (0.57) GPBAR1LMNAKMT2AGAAMEN1
SCHEMBL8408128 0.84 ALDH1A1 (0.60) GPBAR1LMNAKMT2AGAAMEN1
SCHEMBL4721200 0.84 LMNA (0.72) GPBAR1LMNAKMT2AGAAMEN1
SCHEMBL2471701 0.83 GPBAR1 (0.54) GPBAR1LMNAKMT2AGAAMEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-103201268-A Novel piperazine analogs as broad-spectrum influenza antivirals BRISTOL MYERS SQUIBB CO 2013-07-10 CN disclosed