SCHEMBL27913675

SCHEMBL27913675

CCc1cc(OC)cnc1OCC(F)(F)F

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PTGS2 P35354 2/20 0.39
ALDH1A1 P00352 1/20 0.35
MAPT P10636 1/20 0.35
CYP11B1 P15538 1/20 0.35
CYP11B2 P19099 1/20 0.35
PDK2 Q15119 1/20 0.34
PTGS1 P23219 1/20 0.34
CYP17A1 P05093 1/20 0.34
LMNA P02545 2/20 0.33
TRPV1 Q8NER1 1/20 0.33
CYP1A2 P05177 1/20 0.33
CYP2C9 P11712 1/20 0.33
SGK1 O00141 1/20 0.32
SCN9A Q15858 1/20 0.32
CNR2 P34972 1/20 0.32
HDAC3 O15379 1/20 0.32
HDAC1 Q13547 1/20 0.32
HDAC2 Q92769 1/20 0.32
HDAC6 Q9UBN7 1/20 0.32
MEN1 O00255 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL27931866 0.81 CYP11B1 (0.39) PTGS2ALDH1A1MAPTCYP11B1CYP11B2
SCHEMBL16838822 0.81 PTGS2 (0.38) PTGS2ALDH1A1MAPTCYP11B1CYP11B2
SCHEMBL27913649 0.81 CYP11B1 (0.39) PTGS2ALDH1A1MAPTCYP11B1CYP11B2
SCHEMBL27913679 0.81 PTGS2 (0.37) PTGS2ALDH1A1MAPTCYP11B1CYP11B2
SCHEMBL19430888 0.79 LMNA (0.41) PTGS2ALDH1A1LMNACYP1A2CYP2C9
SCHEMBL27913663 0.78 MAPT (0.32) ALDH1A1MAPTCYP17A1SCN9AMEN1
SCHEMBL2715083 0.77 PTGS2 (0.38) PTGS2ALDH1A1MAPTLMNACNR2
SCHEMBL4550333 0.77 PTGS2 (0.38) PTGS2ALDH1A1MAPTCYP17A1CYP1A2
SCHEMBL2715192 0.77 PTGS2 (0.40) PTGS2MAPTPTGS1LMNACNR2
SCHEMBL2716361 0.77 NOTUM (0.41) PTGS2ALDH1A1MAPTLMNASCN9A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-103249721-A Arylamine Derivatives as TTX-S Blockers RAQUALIA PHARMA INC 2013-08-14 CN disclosed