SCHEMBL27929345

SCHEMBL27929345

Nc1cccc(C(=O)NCc2cccc(C(F)(F)F)c2)c1N

nearest known ligand 0.66

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HPGD P15428 3/20 0.61
LMNA P02545 1/20 0.61
MLYCD O95822 1/20 0.60
MEN1 O00255 2/20 0.58
KMT2A Q03164 2/20 0.58
PLA2G1B P04054 1/20 0.58
CYP1A2 P05177 1/20 0.58
CYP3A4 P08684 1/20 0.58
GAA P10253 1/20 0.58
CYP2D6 P10635 1/20 0.58
CYP2C19 P33261 1/20 0.58
TDP1 Q9NUW8 1/20 0.58
ATG4B Q9Y4P1 1/20 0.58
KDM4E B2RXH2 2/20 0.54
ALDH1A1 P00352 2/20 0.54
HSD17B10 Q99714 1/20 0.54
MAPK14 Q16539 1/20 0.54
CCR1 P32246 6/20 0.53
NSD2 O96028 1/20 0.51
PTGS1 P23219 1/20 0.51

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL23864576 0.82 KMT2A (0.66) HPGDLMNAMLYCDMEN1KMT2A
SCHEMBL923670 0.81 LMNA (0.58) HPGDLMNAMLYCDMEN1KMT2A
SCHEMBL24713109 0.80 MLYCD (0.67) HPGDLMNAMLYCDMEN1KMT2A
SCHEMBL3853133 0.80 CCR1 (0.62) HPGDLMNAMLYCDMEN1KMT2A
SCHEMBL5227678 0.78 MLYCD (0.86) HPGDLMNAMLYCDMEN1KMT2A
SCHEMBL23447721 0.78 MLYCD (0.77) HPGDLMNAMLYCDMEN1KMT2A
SCHEMBL1052230 0.78 MLYCD (0.63) HPGDLMNAMLYCDMEN1KMT2A
SCHEMBL31173731 0.78 MLYCD (0.63) HPGDLMNAMLYCDMEN1KMT2A
SCHEMBL26625392 0.78 LMNA (0.69) HPGDLMNAMLYCDMEN1KMT2A
SCHEMBL10491484 0.78 KMT2A (0.67) HPGDLMNAMLYCDMEN1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-103435562-B 6-replaces Benzodiazepine-2,4-cyclohexadione compounds and uses thereof EAST CHINA UNIVERSITY OF SCIENCE AND TECHNOLOGY (CN) 2016-02-24 CN disclosed
CN-103435562-A 6-substituted benzodiazepine-2,4-diketone compound and application thereof UNIV EAST CHINA SCIENCE & TECH 2013-12-11 CN disclosed