SCHEMBL27931908

SCHEMBL27931908

COc1ccc(OCC(C)(F)F)nc1

nearest known ligand 0.41

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
HDAC1 Q13547 1/20 0.41
HDAC8 Q9BY41 1/20 0.41
HDAC6 Q9UBN7 1/20 0.41
HDAC5 Q9UQL6 1/20 0.41
L3MBTL1 Q9Y468 1/20 0.41
DGAT1 O75907 4/20 0.40
TRPV1 Q8NER1 1/20 0.36
TSHR P16473 1/20 0.35
SMN1; SMN2 Q16637 1/20 0.35
LMNA P02545 1/20 0.35
LIPE Q05469 1/20 0.34
HAO1 Q9UJM8 1/20 0.34
KDM4E B2RXH2 1/20 0.34
POLB P06746 1/20 0.34
RAB9A P51151 1/20 0.34
CHRNB2 P17787 1/20 0.34
CHRNA4 P43681 1/20 0.34
NFE2L2 Q16236 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL27931886 0.82 HDAC1 (0.39) HDAC1HDAC8HDAC6HDAC5L3MBTL1
SCHEMBL19767298 0.79 L3MBTL1 (0.42) HDAC6L3MBTL1DGAT1KDM4EPOLB
SCHEMBL28806907 0.78 SCN5A (0.46) HDAC1HDAC8HDAC6HDAC5
SCHEMBL7909762 0.77 RUNX1 (0.40) HDAC1HDAC8HDAC6HDAC5L3MBTL1
SCHEMBL3816388 0.75 NNMT (0.48) L3MBTL1LMNAHAO1KDM4ECHRNB2
SCHEMBL29525223 0.75 NNMT (0.48) L3MBTL1LMNAHAO1KDM4ECHRNB2
SCHEMBL2714106 0.75 L3MBTL1 (0.43) L3MBTL1DGAT1TRPV1POLB
SCHEMBL4550334 0.75 L3MBTL1 (0.40) L3MBTL1DGAT1POLB
SCHEMBL27775336 0.74 KDM4E (0.41) SMN1; SMN2HAO1KDM4EPOLBRAB9A
SCHEMBL27988925 0.74 L3MBTL1 (0.45) L3MBTL1TSHRSMN1; SMN2LMNAKDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-103249721-A Arylamine Derivatives as TTX-S Blockers RAQUALIA PHARMA INC 2013-08-14 CN disclosed