SCHEMBL279333

SCHEMBL279333

C=C(/N=C/c1cc(I)ccc1OCC1CCN(C(=O)OC(C)(C)C)CC1)O[Si](C)(C)C

nearest known ligand 0.45

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
GPR119 Q8TDV5 13/20 0.40
CHEK2 O96017 1/20 0.40
CSF1R P07333 1/20 0.39
ALOX5AP P20292 1/20 0.38
FEN1 P39748 1/20 0.38
FAAH O00519 1/20 0.38
SLC2A1 P11166 1/20 0.37
KDM4E B2RXH2 1/20 0.36
PKM P14618 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL279337 0.88 PDE4B (0.44) GPR119CHEK2
SCHEMBL279312 0.85 PIK3CD (0.44) GPR119
SCHEMBL275719 0.82 CHEK2 (0.44) GPR119CHEK2CSF1RALOX5APFEN1
SCHEMBL275711 0.80 PDE4B (0.38) GPR119
SCHEMBL279410 0.80 PDE4B (0.38) GPR119
SCHEMBL279056 0.78 PDE4B (0.44) GPR119CHEK2
SCHEMBL279069 0.76 GPR119 (0.44) GPR119
SCHEMBL278898 0.75 PIK3CD (0.44) GPR119
SCHEMBL279147 0.72 HPGD (0.32)
SCHEMBL15539222 0.71 PTGDR2 (0.46) GPR119CHEK2CSF1RALOX5APFEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8134001-B2 Spiroindolinone derivatives HOFFMANN-LA ROCHE INC. (US) 2012-03-13 US disclosed
US-20090156610-A1 Spiroindolinone Derivatives DING QINGJIE 2009-06-18 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20090156610-A1 Spiroindolinone Derivatives SDHA, AR, XPOT GPR119 2589/4885CHEK2 688/4885CSF1R 3130/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.