SCHEMBL27936014

SCHEMBL27936014

Cc1cnc2c(C(=O)C=O)c(C)ccc2c1

nearest known ligand 0.53

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
CCR1 P32246 2/20 0.53
CCR5 P51681 2/20 0.53
CCR8 P51685 2/20 0.53
PARP1 P09874 2/20 0.46
KDM4E B2RXH2 1/20 0.44
PSMD14 O00487 2/20 0.41
COPS5 Q92905 2/20 0.41
NFKBIA P25963 1/20 0.36
SLC40A1 Q9NP59 4/20 0.35
CYP1A2 P05177 1/20 0.34
EGLN3 Q9H6Z9 1/20 0.32
ALK Q9UM73 1/20 0.32
PADI4 Q9UM07 2/20 0.32
SLC16A3 O15427 1/20 0.31
STAMBP O95630 1/20 0.31
ABL1 P00519 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13620452 0.83 CCR1 (0.58) CCR1CCR5CCR8PARP1KDM4E
SCHEMBL28189404 0.77 LMNA (0.51) CCR1CCR5CCR8PARP1KDM4E
SCHEMBL27925228 0.72 CCR1 (0.45) CCR1CCR5CCR8PARP1KDM4E
SCHEMBL30492603 0.72 CCR1 (1.00) CCR1CCR5CCR8PARP1KDM4E
SCHEMBL686948 0.72 CCR1 (1.00) CCR1CCR5CCR8PARP1KDM4E
SCHEMBL862768 0.72 CCR1 (0.73) CCR1CCR5CCR8PARP1KDM4E
SCHEMBL862480 0.71 CCR1 (0.72) CCR1CCR5CCR8PARP1KDM4E
Quinmerac SCHEMBL29433226 0.71 ALK (0.60) CCR1CCR5CCR8PARP1KDM4E
Quinmerac SCHEMBL8539662 0.71 ALK (0.60) CCR1CCR5CCR8PARP1KDM4E
Quinmerac SCHEMBL29351452 0.71 ALK (0.60) CCR1CCR5CCR8PARP1KDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-103534238-B Total synthesis of redox active 1, 4-naphthoquinones and their metabolites and their therapeutic use as antimalarial and schistosomimetics 国家科研中心 2018-01-02 CN disclosed
CN-103534238-A Total synthesis of redox active 1, 4-naphthoquinones and their metabolites and their therapeutic use as antimalarial and schistosomimetics CENTRE NAT RECH SCIENT 2014-01-22 CN disclosed