SCHEMBL28189404

SCHEMBL28189404

Cc1ccc2cccnc2c1C(=O)C=O

nearest known ligand 0.51

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
LMNA P02545 3/20 0.51
ERN1 O75460 1/20 0.46
CCR1 P32246 4/20 0.46
CCR8 P51685 4/20 0.46
CCR5 P51681 3/20 0.46
TDP1 Q9NUW8 3/20 0.46
MAPT P10636 3/20 0.46
KDM4E B2RXH2 2/20 0.46
HTT P42858 2/20 0.46
SMN1; SMN2 Q16637 2/20 0.46
TP53 P04637 2/20 0.46
MMP2 P08253 2/20 0.46
TSHR P16473 2/20 0.46
GMNN O75496 1/20 0.46
HSP90AA1 P07900 1/20 0.46
CYP3A4 P08684 1/20 0.46
CYP2D6 P10635 1/20 0.46
MMP9 P14780 1/20 0.46
ALOX15 P16050 1/20 0.46
NFKB1 P19838 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11430231 0.82 LMNA (0.56) LMNACCR1CCR8CCR5TDP1
SCHEMBL28324949 0.82 CCR1 (0.47) LMNAERN1CCR1CCR8CCR5
SCHEMBL28264597 0.81 ERN1 (0.46) LMNAERN1CCR1CCR8CCR5
SCHEMBL28263607 0.81 ERN1 (0.46) LMNAERN1CCR1CCR8CCR5
SCHEMBL9945612 0.78 LMNA (0.51) LMNACCR1CCR8CCR5TDP1
SCHEMBL9944365 0.78 LMNA (0.47) LMNACCR1CCR8CCR5TDP1
SCHEMBL27936014 0.77 CCR1 (0.53) CCR1CCR8CCR5KDM4ESLC40A1
SCHEMBL28581006 0.74 KDM4E (0.46) LMNAERN1CCR1CCR8CCR5
SCHEMBL20669627 0.73 ERN1 (0.65) LMNAERN1CCR1CCR8CCR5
SCHEMBL27489489 0.73 PARP1 (0.64) LMNAERN1CCR1CCR8CCR5

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-103534238-B Total synthesis of redox active 1, 4-naphthoquinones and their metabolites and their therapeutic use as antimalarial and schistosomimetics 国家科研中心 2018-01-02 CN disclosed