SCHEMBL27945232

SCHEMBL27945232

CC(C)(C)C(=O)ON1CCC(c2ccc3[nH]ncc3c2)CC1

nearest known ligand 0.48

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
FASN P49327 1/20 0.48
CCNC P24863 1/20 0.42
CDK8 P49336 1/20 0.42
SLC6A2 P23975 3/20 0.41
SLC6A4 P31645 3/20 0.41
SLC6A3 Q01959 3/20 0.41
ROCK2 O75116 7/20 0.41
CYP3A4 P08684 3/20 0.41
POLB P06746 1/20 0.40
ROCK1 Q13464 1/20 0.39
PRMT5 O14744 2/20 0.39
PIK3CD O00329 1/20 0.39
PLK4 O00444 1/20 0.38
HSD11B1 P28845 2/20 0.38
CYP2D6 P10635 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL27774785 0.90 SLC6A2 (0.44) FASNCCNCCDK8SLC6A2SLC6A4
SCHEMBL9952336 0.83 FASN (0.52) FASNROCK2CYP3A4PIK3CD
SCHEMBL27665777 0.81 CYP3A4 (0.57) CDK8SLC6A2SLC6A4SLC6A3ROCK2
SCHEMBL15556237 0.78 FASN (0.55) FASNCCNCCDK8ROCK2CYP3A4
SCHEMBL9917339 0.78 SLC6A2 (0.55) FASNSLC6A2SLC6A4SLC6A3ROCK2
SCHEMBL27926231 0.76 TLR7 (0.36) CCNCCDK8
SCHEMBL3328409 0.76 PIK3CD (0.49) FASNCCNCCDK8SLC6A2SLC6A4
SCHEMBL4833473 0.75 ROCK2 (0.52) FASNSLC6A2SLC6A4SLC6A3ROCK2
SCHEMBL27984917 0.75 HSD11B1 (0.46) ROCK2HSD11B1
SCHEMBL27792727 0.74 CYP3A4 (0.47) ROCK2CYP3A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-103429585-A Indazolyl triazole derivatives as interleukin-1 receptor associated kinase inhibitors MERCK SERONO SA 2013-12-04 CN disclosed