SCHEMBL27946366

SCHEMBL27946366

Nc1ncc(Br)cc1N1CCc2ccccc2C1=O

nearest known ligand 0.45

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
BCAT2 O15382 2/20 0.45
GRM4 Q14833 1/20 0.43
TDP1 Q9NUW8 1/20 0.38
L3MBTL1 Q9Y468 1/20 0.38
CYP11B2 P19099 2/20 0.37
CYP11B1 P15538 1/20 0.37
GRM1 Q13255 1/20 0.37
GRIN2D O15399 1/20 0.36
GRIN3B O60391 1/20 0.36
GRIN1 Q05586 1/20 0.36
GRIN2A Q12879 1/20 0.36
GRIN2B Q13224 1/20 0.36
GRIN2C Q14957 1/20 0.36
GRIN3A Q8TCU5 1/20 0.36
AOC3 Q16853 2/20 0.36
MAP3K14 Q99558 1/20 0.36
SMN1; SMN2 Q16637 3/20 0.36
NPC1 O15118 2/20 0.36
RAB9A P51151 2/20 0.36
MAPT P10636 2/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL19812980 0.77 MAPK1 (0.48) BCAT2GRM4
SCHEMBL4088660 0.76 KMT2A (0.44) CYP11B2CYP11B1MAP3K14SMN1; SMN2NPC1
SCHEMBL16914120 0.71 HSD17B10 (0.49) L3MBTL1CYP11B2NPC1HTTHPGD
SCHEMBL123331 0.69 BCAT2 (0.45) BCAT2TDP1GRM1NPC1RAB9A
SCHEMBL23356622 0.69 KMT2A (0.55) BCAT2TDP1GRM1SMN1; SMN2NPC1
SCHEMBL29458437 0.69 KMT2A (0.55) BCAT2TDP1GRM1SMN1; SMN2NPC1
SCHEMBL29163638 0.69 CRBN (0.56) BCAT2GRM4GRIN2DGRIN3BGRIN1
SCHEMBL798870 0.68 CYP11B2 (0.47) BCAT2GRM4TDP1CYP11B2CYP11B1
SCHEMBL29923615 0.68 CYP11B2 (0.50) BCAT2CYP11B2CYP11B1
SCHEMBL2600444 0.68 NPC1 (0.68) BCAT2CYP11B2CYP11B1AOC3SMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-103429582-A MST1 kinase inhibitors and method of use thereof LEXICON PHARMACEUTICALS INC 2013-12-04 CN disclosed