SCHEMBL27947482

SCHEMBL27947482

c1cnc2[nH]nc(-c3cncnc3)c2c1

nearest known ligand 0.50

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
IDO1 P14902 1/20 0.50
LRRK2 Q5S007 1/20 0.50
PIM1 P11309 10/20 0.47
CYP2A6 P11509 2/20 0.46
PIM2 Q9P1W9 2/20 0.43
PIM3 Q86V86 1/20 0.43
CLK2 P49760 3/20 0.43
DYRK1A Q13627 3/20 0.43
CLK3 P49761 2/20 0.43
MAP2K4 P45985 1/20 0.42
AXL P30530 1/20 0.41
GRM4 Q14833 1/20 0.41
WNT1 P04628 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2926259 0.82 PIM1 (0.51) IDO1LRRK2PIM1PIM2PIM3
SCHEMBL1513056 0.80 ALDH1A1 (0.55) IDO1LRRK2PIM1PIM2PIM3
SCHEMBL30931548 0.80 ALDH1A1 (0.55) IDO1LRRK2PIM1PIM2PIM3
SCHEMBL17922026 0.78 LRRK2 (0.41) IDO1LRRK2PIM1CYP2A6PIM2
SCHEMBL29930912 0.78 MAPK1 (0.42) IDO1LRRK2PIM1DYRK1A
SCHEMBL25029271 0.76 ALDH1A1 (0.54) PIM1MAP2K4GRM4
SCHEMBL9877148 0.76 PDPK1 (0.49) IDO1LRRK2MAP2K4
SCHEMBL10452107 0.74 LRRK2 (0.62) IDO1LRRK2MAP2K4GRM4
SCHEMBL1639739 0.74 LRRK2 (0.67) IDO1LRRK2PIM1CYP2A6PIM2
SCHEMBL18449016 0.74 CLK2 (0.61) CLK2DYRK1ACLK3WNT1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-105503862-B Inhibitors of influenza viruses replication 沃泰克斯药物股份有限公司 2018-02-02 CN disclosed
CN-103492381-A Inhibitors of influenza virus replication VERTEX PHARMA 2014-01-01 CN disclosed