SCHEMBL9877148

SCHEMBL9877148

Oc1ccc(-c2n[nH]c3ncccc23)cc1

nearest known ligand 0.49

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PDPK1 O15530 1/20 0.49
HSP90AB1 P08238 1/20 0.49
MAPK1 P28482 3/20 0.47
MAP2K4 P45985 3/20 0.47
MAPKAPK2 P49137 3/20 0.47
MAPK6 Q16659 3/20 0.47
RIPK1 Q13546 3/20 0.47
MAPKAPK3 Q16644 2/20 0.47
MAPKAPK5 Q8IW41 1/20 0.47
FGFR1 P11362 2/20 0.47
FGFR2 P21802 2/20 0.47
FGFR3 P22607 1/20 0.47
ROCK1 Q13464 1/20 0.41
CDC7 O00311 1/20 0.41
GAA P10253 2/20 0.40
CHEK1 O14757 3/20 0.39
IDO1 P14902 2/20 0.39
LRRK2 Q5S007 1/20 0.39
CCNB2 O95067 1/20 0.39
CDK1 P06493 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1513056 0.84 ALDH1A1 (0.55) GAAIDO1LRRK2NPSR1KDM4E
SCHEMBL30931548 0.84 ALDH1A1 (0.55) GAAIDO1LRRK2NPSR1KDM4E
SCHEMBL25029271 0.83 ALDH1A1 (0.54) MAPK1MAP2K4CDC7GSK3BALDH1A1
SCHEMBL2926259 0.82 PIM1 (0.51) PDPK1MAPK1ROCK1GAAIDO1
SCHEMBL17922026 0.78 LRRK2 (0.41) ROCK1GAAIDO1LRRK2KDM4E
SCHEMBL27947482 0.76 IDO1 (0.50) MAP2K4IDO1LRRK2
SCHEMBL1573790 0.76 AXL (0.41) HSP90AB1CDC7IDO1LRRK2GSK3A
SCHEMBL29930484 0.75 DYRK1B (0.56) PDPK1HSP90AB1MAPK1MAP2K4MAPKAPK2
SCHEMBL22044852 0.74 ROCK1 (0.62) ROCK1GAA
SCHEMBL10530840 0.74 CA1 (0.43) GAA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5006520-A Antibiotics, antitumor agents, treatment of blood disorders YOSHITOMI PHARMACEUTICAL INDUSTRIES, LTD. (JP) 1991-04-09 US disclosed
EP-0338087-A1 FUSED PYRAZOLE COMPOUNDS, PROCESS FOR THEIR PREPARATION, AND THEIR MEDICINAL USE Yoshitomi Pharmaceutical Industries, Ltd. (JP) 1989-10-25 EP disclosed