SCHEMBL27947728

SCHEMBL27947728

COc1cc(N)cc(C(=O)OC(C)(C)C)c1N

nearest known ligand 0.44

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 3/20 0.44
POLB P06746 1/20 0.44
ALDH1A1 P00352 1/20 0.42
GAA P10253 1/20 0.36
HTT P42858 1/20 0.35
MTNR1A P48039 3/20 0.34
MTNR1B P49286 3/20 0.34
GRM6 O15303 1/20 0.34
EGFR P00533 1/20 0.34
NFKB1 P19838 1/20 0.34
NFKB2 Q00653 1/20 0.34
RELA Q04206 1/20 0.34
CREBBP Q92793 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1100205 0.81 ALDH1A1 (0.63) KDM4EALDH1A1GAAHTT
SCHEMBL5428749 0.78 ALDH1A1 (0.62) KDM4EPOLBALDH1A1HTT
SCHEMBL27996077 0.74 CA12 (0.42) KDM4EPOLBALDH1A1GAAGRM6
SCHEMBL31656211 0.73 CYP3A4 (0.55) KDM4EPOLBALDH1A1GAAEGFR
SCHEMBL2616107 0.73 CYP3A4 (0.55) KDM4EPOLBALDH1A1GAAEGFR
SCHEMBL31188292 0.73 ALDH1A1 (0.49) KDM4EALDH1A1GAAGRM6
SCHEMBL28309007 0.72 CYP3A4 (0.40) KDM4EGAAGRM6EGFR
SCHEMBL28362778 0.72 ACHE (0.48) KDM4EPOLBALDH1A1GAAMTNR1A
SCHEMBL1185611 0.71 KMT2A (0.52) KDM4EPOLBALDH1A1GAAGRM6
SCHEMBL28903578 0.71 HTT (0.59) KDM4EALDH1A1HTTMTNR1AMTNR1B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-103501612-A Compounds for inhibiting cell proliferation in EGFR-driven cancers ARIAD PHARMA INC 2014-01-08 CN disclosed