SCHEMBL27951093

SCHEMBL27951093

CC(C)(C)OC(=O)NCC(=O)N[C@@H](Cc1c[nH]c2ccccc12)C(=O)OCc1ccccc1

nearest known ligand 0.71

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TACR1 P25103 13/20 0.71
ACE P12821 1/20 0.61
KLK7 P49862 1/20 0.61
CTSL P07711 1/20 0.59
CTSS P25774 1/20 0.59
CTSK P43235 1/20 0.59
LNPEP Q9UIQ6 1/20 0.59
IL1RN P18510 1/20 0.59
ERAP2 Q6P179 1/20 0.59
ERAP1 Q9NZ08 1/20 0.59
KDM4E B2RXH2 1/20 0.57
MEN1 O00255 1/20 0.57
ALDH1A1 P00352 1/20 0.57
LMNA P02545 1/20 0.57
TP53 P04637 1/20 0.57
CYP1A2 P05177 1/20 0.57
POLB P06746 1/20 0.57
CYP3A4 P08684 1/20 0.57
CYP2D6 P10635 1/20 0.57
MAPT P10636 1/20 0.57

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL27951096 1.00 TACR1 (0.71) TACR1ACEKLK7CTSLCTSS
SCHEMBL29397912 0.91 TACR1 (0.82) TACR1ACEKLK7CTSLCTSS
SCHEMBL16464197 0.91 TACR1 (0.82) TACR1ACEKLK7CTSLCTSS
SCHEMBL8697113 0.91 TACR1 (0.82) TACR1ACEKLK7CTSLCTSS
SCHEMBL5355362 0.91 TACR1 (0.82) TACR1ACEKLK7CTSLCTSS
SCHEMBL29419166 0.90 TACR1 (0.65) TACR1ACECTSLCTSSCTSK
SCHEMBL31465284 0.89 ACE (0.69) TACR1ACECTSLCTSSCTSK
SCHEMBL27902201 0.89 ACE (0.69) TACR1ACECTSLCTSSCTSK
SCHEMBL27902203 0.89 ACE (0.69) TACR1ACECTSLCTSSCTSK
SCHEMBL29194048 0.88 MAPT (0.67) TACR1ACEKLK7CTSLCTSS

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-102807601-B Aminoacyl-tryptophanyl-5-methoxytryptamine and preparation method and application thereof UNIV CAPITAL MEDICAL SCIENCES 2014-02-26 CN disclosed
CN-102807601-A Aminoacyl-tryptophanyl-5-methoxytryptamine and preparation method and application thereof UNIV CAPITAL MEDICAL 2012-12-05 CN disclosed