SCHEMBL27902201

SCHEMBL27902201

CC(C)(C)OC(=O)NCC(=O)N[C@@H](Cc1c[nH]c2ccccc12)C(=O)O

nearest known ligand 0.69

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ACE P12821 5/20 0.69
CTSL P07711 1/20 0.65
CTSS P25774 1/20 0.65
CTSK P43235 1/20 0.65
SCN9A Q15858 1/20 0.61
KDM4E B2RXH2 1/20 0.60
TACR1 P25103 2/20 0.59
POLB P06746 3/20 0.59
TP53 P04637 2/20 0.59
P2RY14 Q15391 1/20 0.59
ALOX15 P16050 1/20 0.59
HDAC3 O15379 2/20 0.58
HDAC4 P56524 2/20 0.58
HDAC1 Q13547 2/20 0.58
HDAC7 Q8WUI4 2/20 0.58
HDAC2 Q92769 2/20 0.58
HDAC10 Q969S8 2/20 0.58
HDAC11 Q96DB2 2/20 0.58
HDAC8 Q9BY41 2/20 0.58
HDAC6 Q9UBN7 2/20 0.58

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL31465284 1.00 ACE (0.69) ACECTSLCTSSCTSKSCN9A
SCHEMBL27902203 1.00 ACE (0.69) ACECTSLCTSSCTSKSCN9A
SCHEMBL29419166 0.91 TACR1 (0.65) ACECTSLCTSSCTSKTACR1
SCHEMBL30568723 0.90 ACE (0.73) ACECTSLCTSSCTSKSCN9A
SCHEMBL16672124 0.89 ALOX15 (0.64) ACEKDM4EPOLBTP53P2RY14
SCHEMBL850438 0.89 ACE (0.77) ACECTSLCTSSCTSKSCN9A
SCHEMBL29367687 0.89 ACE (0.77) ACECTSLCTSSCTSKSCN9A
SCHEMBL1486167 0.89 ACE (0.77) ACECTSLCTSSCTSKSCN9A
SCHEMBL30976323 0.89 ACE (0.77) ACECTSLCTSSCTSKSCN9A
SCHEMBL1003555 0.89 ACE (0.77) ACECTSLCTSSCTSKSCN9A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-102807601-B Aminoacyl-tryptophanyl-5-methoxytryptamine and preparation method and application thereof UNIV CAPITAL MEDICAL SCIENCES 2014-02-26 CN disclosed
CN-102807601-A Aminoacyl-tryptophanyl-5-methoxytryptamine and preparation method and application thereof UNIV CAPITAL MEDICAL 2012-12-05 CN disclosed