SCHEMBL27959751

SCHEMBL27959751

NC(=O)NC(c1ccccn1)c1ccccn1

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
S1PR2 O95136 1/20 0.46
S1PR4 O95977 1/20 0.46
S1PR3 Q99500 1/20 0.46
LMNA P02545 2/20 0.45
CYP1A2 P05177 2/20 0.42
CYP3A4 P08684 2/20 0.42
GAA P10253 2/20 0.42
ALDH1A1 P00352 4/20 0.42
SLC6A3 Q01959 2/20 0.41
SLC6A2 P23975 1/20 0.41
SLC6A4 P31645 1/20 0.41
KDM4E B2RXH2 2/20 0.41
NPC1 O15118 1/20 0.40
PKM P14618 1/20 0.40
RAB9A P51151 1/20 0.40
ABCB11 O95342 1/20 0.40
ESR1 P03372 1/20 0.40
ADRA2A P08913 1/20 0.40
CYP2C9 P11712 1/20 0.40
TSHR P16473 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29029999 0.86 S1PR2 (0.44) S1PR2S1PR4S1PR3LMNACYP1A2
SCHEMBL2339352 0.83 S1PR2 (0.50) S1PR2S1PR4S1PR3LMNACYP1A2
SCHEMBL9750150 0.82 CYP1A2 (0.47) CYP1A2CYP3A4ALDH1A1
SCHEMBL438354 0.76 CYP1A2 (0.47) LMNACYP1A2CYP3A4GAAALDH1A1
SCHEMBL7517110 0.73 SLC6A2 (0.52) S1PR2S1PR4S1PR3LMNACYP1A2
Carbamic Acid SCHEMBL11335902 0.73 KDM4E (0.51) LMNACYP1A2CYP3A4GAAALDH1A1
SCHEMBL6796070 0.73 KDM4E (0.47) LMNACYP1A2CYP3A4GAAALDH1A1
SCHEMBL20993625 0.73 CYP1A2 (0.45) LMNACYP1A2CYP3A4GAAALDH1A1
SCHEMBL20993622 0.73 CYP1A2 (0.45) LMNACYP1A2CYP3A4GAAALDH1A1
SCHEMBL2656952 0.73 CYP1A2 (0.45) LMNACYP1A2CYP3A4GAAALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-103922998-A Heterodimers Of Glutamic Acid MOLECULAR INSIGHT PHARM INC 2014-07-16 CN disclosed
CN-101778910-B Heterodimers of glutamic acid MOLECULAR INSIGHT PHARM INC 2014-05-28 CN disclosed