SCHEMBL27973449

SCHEMBL27973449

NC(=O)c1ccc2c(c1)C=CCN2

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TSHR P16473 1/20 0.38
SIRT2 Q8IXJ6 1/20 0.38
LCK P06239 1/20 0.36
PARP1 P09874 6/20 0.34
MAPKAPK2 P49137 2/20 0.33
IP6K1 Q92551 1/20 0.33
RPS6KA3 P51812 1/20 0.33
MAPK1 P28482 1/20 0.33
MAP2K4 P45985 1/20 0.33
MAPKAPK3 Q16644 1/20 0.33
MAPK6 Q16659 1/20 0.33
MAPKAPK5 Q8IW41 1/20 0.33
PKN1 Q16512 1/20 0.33
PKN2 Q16513 1/20 0.33
PARP15 Q460N3 2/20 0.33
PARP14 Q460N5 2/20 0.33
PARP10 Q53GL7 2/20 0.33
ALDH1A1 P00352 2/20 0.33
TNKS O95271 1/20 0.33
TNKS2 Q9H2K2 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL12482950 0.85 KDM4E (0.45) TSHRSIRT2MAPK1ALDH1A1KDM4E
SCHEMBL2115737 0.75 SIRT2 (0.37) TSHRSIRT2LCKPARP1MAPKAPK2
SCHEMBL28259357 0.75 KDM4E (0.41) TSHRSIRT2MAPK1ALDH1A1KDM4E
SCHEMBL1007936 0.71 LCK (0.37) TSHRSIRT2LCKPARP1IP6K1
SCHEMBL6033497 0.71 MEN1 (0.39) ALDH1A1SMN1; SMN2KMT2A
SCHEMBL22418394 0.71 ADORA3 (0.36) TSHRLCKKMT2A
SCHEMBL30445575 0.71 NNMT (0.51) SIRT2SMN1; SMN2
SCHEMBL5579532 0.71 TSHR (0.44) TSHRSIRT2LCKPARP1RPS6KA3
SCHEMBL4437948 0.71 TSHR (0.44) TSHRSIRT2LCKPARP1MAPKAPK2
SCHEMBL20568616 0.70 BTK (0.32) LCK

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-110430878-A Antitumor agent and bromine structural domain inhibitor FUJIFILM CORP 2019-11-08 CN disclosed
CN-108137505-A Nitrogen-containing heterocycle compound 富士胶片株式会社 2018-06-08 CN disclosed
CN-104039152-A Antibacterial compounds GLAXO GROUP LTD 2014-09-10 CN disclosed