SCHEMBL27974841

SCHEMBL27974841

[CH2]Cc1cn2ncnc(N)c2c1-c1ccc(N)c(Cl)c1

nearest known ligand 0.38

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
ACVRL1 P37023 1/20 0.38
ALDH1A1 P00352 1/20 0.36
CYP3A4 P08684 1/20 0.36
TSHR P16473 1/20 0.36
MAPK1 P28482 1/20 0.36
FGFR1 P11362 17/20 0.35
ESR2 Q92731 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL27663138 0.86 ACVRL1 (0.37) ACVRL1FGFR1
SCHEMBL27974840 0.84 TP53 (0.36) ACVRL1ALDH1A1CYP3A4TSHRMAPK1
SCHEMBL27682734 0.82 FGFR1 (0.36) FGFR1
SCHEMBL763960 0.81 FGFR1 (0.42) FGFR1
SCHEMBL27663275 0.78 KMT2A (0.42) ALDH1A1CYP3A4FGFR1
SCHEMBL27663264 0.74 KDR (0.45) MAPK1FGFR1
SCHEMBL761901 0.74 FGFR1 (0.36) ALDH1A1CYP3A4TSHRMAPK1FGFR1
SCHEMBL742983 0.74 EGFR (0.46) ALDH1A1FGFR1
SCHEMBL27682729 0.73 KDR (0.44) MAPK1FGFR1
SCHEMBL28761004 0.72 RIPK1 (0.53)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-101820762-B Pyrrolotriazine derivatives for treating cancer through inhibition of aurora kinase BAYER HEALTHCARE LLC 2014-07-30 CN disclosed