SCHEMBL27978468

SCHEMBL27978468

CCOC(C1CCN(c2ncc3c(-c4ccccc4)c(NC(=O)C(C)C)sc3n2)CC1)N1CCCC1

nearest known ligand 0.56

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PTPN11 Q06124 6/20 0.37
HPGD P15428 3/20 0.35
ALDH1A1 P00352 2/20 0.35
POLB P06746 2/20 0.35
SMN1; SMN2 Q16637 2/20 0.35
KDM4E B2RXH2 1/20 0.35
MEN1 O00255 1/20 0.35
CYP2C9 P11712 1/20 0.35
CYP2C19 P33261 1/20 0.35
HTT P42858 1/20 0.35
KMT2A Q03164 1/20 0.35
NPSR1 Q6W5P4 1/20 0.35
TP53 P04637 1/20 0.35
THRB P10828 1/20 0.35
GLS O94925 3/20 0.34
MAPT P10636 2/20 0.33
CPT2 P23786 1/20 0.33
CPT1A P50416 1/20 0.33
P2RY12 Q9H244 1/20 0.33
RAB9A P51151 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL27978490 0.92 PTPN11 (0.38) PTPN11HPGDALDH1A1POLBSMN1; SMN2
SCHEMBL27978780 0.91 MAPT (0.37) PTPN11HPGDALDH1A1POLBSMN1; SMN2
SCHEMBL14965244 0.81 HTR1A (0.38) KDM4E
SCHEMBL27978487 0.80 PTPN11 (0.33) PTPN11HPGDALDH1A1MEN1CYP2C9
SCHEMBL27978494 0.77 SMN1; SMN2 (0.39) SMN1; SMN2KDM4EKMT2ATP53
SCHEMBL27978691 0.74 ADRB3 (0.41) MEN1KMT2A
SCHEMBL27978717 0.72 SMN1; SMN2 (0.38) POLBSMN1; SMN2HTTKMT2A
SCHEMBL14965345 0.72 HTR2A (0.36) KDM4E
SCHEMBL27978714 0.71 ELANE (0.34) ALDH1A1MAPT
SCHEMBL27978447 0.70 KMT2A (0.42) HPGDALDH1A1SMN1; SMN2KDM4EMEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-104011054-A Thieno- and furo-pyrimidines and pyridines, useful as potassium channel inhibitors XENTION LTD 2014-08-27 CN disclosed