SCHEMBL27980433

SCHEMBL27980433

ONCc1ccc(-c2nccs2)cn1

nearest known ligand 0.50

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ADRB2 P07550 3/20 0.50
LOXL2 Q9Y4K0 1/20 0.46
CYP2A6 P11509 1/20 0.46
PDPK1 O15530 1/20 0.43
CHEK2 O96017 1/20 0.39
HDAC2 Q92769 2/20 0.36
HDAC3 O15379 1/20 0.36
HDAC4 P56524 1/20 0.36
HDAC1 Q13547 1/20 0.36
HDAC7 Q8WUI4 1/20 0.36
HDAC10 Q969S8 1/20 0.36
HDAC11 Q96DB2 1/20 0.36
HDAC8 Q9BY41 1/20 0.36
HDAC6 Q9UBN7 1/20 0.36
HDAC9 Q9UKV0 1/20 0.36
HDAC5 Q9UQL6 1/20 0.36
PORCN Q9H237 1/20 0.36
PTGDR2 Q9Y5Y4 1/20 0.36
ESR1 P03372 1/20 0.36
SMPD3 Q9NY59 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL16597351 0.82 LOXL2 (0.50) ADRB2LOXL2CYP2A6PDPK1CHEK2
SCHEMBL16610138 0.79 LOXL2 (0.50) ADRB2LOXL2CYP2A6PDPK1CHEK2
SCHEMBL13622938 0.79 ADRB2 (0.50) ADRB2LOXL2CYP2A6PDPK1CHEK2
SCHEMBL13615828 0.75 ADRB2 (0.46) ADRB2LOXL2CYP2A6PDPK1CHEK2
SCHEMBL4355883 0.75 LOXL2 (0.50) ADRB2LOXL2CYP2A6PDPK1CHEK2
SCHEMBL27980432 0.73 CYP2A6 (0.44) ADRB2LOXL2CYP2A6PDPK1CHEK2
SCHEMBL722198 0.71 PDPK1 (0.77) ADRB2LOXL2CYP2A6PDPK1CHEK2
SCHEMBL28790747 0.71 LOXL2 (0.42) ADRB2LOXL2CYP2A6PDPK1CHEK2
SCHEMBL23832336 0.69 CYP2A6 (0.55) ADRB2LOXL2CYP2A6PDPK1CHEK2
SCHEMBL14814093 0.69 CYP2A6 (0.55) ADRB2LOXL2CYP2A6PDPK1CHEK2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-104151381-A Anti-bacterial activity of 9-HYDROXY derivatives of 6, 11-bicyclolides ENANTA PHARM INC 2014-11-19 CN disclosed
CN-102088848-B Antibacterial activity of 6, 11-bicyclic 9-hydroxy derivatives ENANTA PHARM INC 2014-07-30 CN disclosed