SCHEMBL27985359

SCHEMBL27985359

C#Cc1ccc(NC(=O)C(F)(F)F)c(OC)c1

nearest known ligand 0.50

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP1A2 P05177 2/20 0.50
CYP2C9 P11712 1/20 0.50
CYP2C19 P33261 1/20 0.50
TSHR P16473 1/20 0.50
NPSR1 Q6W5P4 1/20 0.50
ABCC9 O60706 1/20 0.44
ABCC8 Q09428 1/20 0.44
KCNJ11 Q14654 1/20 0.44
KCNJ8 Q15842 1/20 0.44
PDK1 Q15118 1/20 0.44
PDK2 Q15119 1/20 0.44
PDK3 Q15120 1/20 0.44
PDK4 Q16654 1/20 0.44
ALDH1A1 P00352 4/20 0.41
LPAR1 Q92633 2/20 0.41
HTT P42858 2/20 0.40
MLYCD O95822 1/20 0.39
CYP1A1 P04798 1/20 0.39
CYP1B1 Q16678 1/20 0.39
ATM Q13315 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3441915 0.89 CYP1A2 (0.54) CYP1A2CYP2C9CYP2C19TSHRNPSR1
SCHEMBL2552734 0.80 TSHR (0.74) CYP1A2CYP2C9CYP2C19TSHRNPSR1
SCHEMBL29785065 0.80 TSHR (0.74) CYP1A2CYP2C9CYP2C19TSHRNPSR1
SCHEMBL6555240 0.78 CYP1A2 (0.54) CYP1A2CYP2C9CYP2C19TSHRNPSR1
SCHEMBL1238843 0.78 CYP1A2 (0.54) CYP1A2CYP2C9CYP2C19TSHRNPSR1
SCHEMBL3539902 0.78 PDK1 (0.40) CYP1A2CYP2C9CYP2C19TSHRPDK1
SCHEMBL6811200 0.78 MAPT (0.54) CYP1A2CYP2C9CYP2C19TSHRNPSR1
SCHEMBL15903926 0.77 ABCC9 (0.58) CYP1A2CYP2C9CYP2C19TSHRNPSR1
SCHEMBL29440834 0.77 ABCC9 (0.58) CYP1A2CYP2C9CYP2C19TSHRNPSR1
SCHEMBL3442075 0.77 MEN1 (0.40) CYP1A2CYP2C9CYP2C19TSHRPDK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-104151292-A Indole derivative or pharmaceutically acceptable salt thereof KISSEI PHARMACEUTICAL 2014-11-19 CN disclosed