SCHEMBL27985451

SCHEMBL27985451

O=C(O)c1ccc(CCBr)c(F)c1F

nearest known ligand 0.38

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 1/20 0.38
ASPH Q12797 1/20 0.38
KDM8 Q8N371 1/20 0.38
CYP1A2 P05177 1/20 0.37
CES2 O00748 2/20 0.35
CES1 P23141 2/20 0.35
FOLH1 Q04609 1/20 0.34
PTPN1 P18031 2/20 0.33
DCLRE1B Q9H816 1/20 0.33
ALB P02768 1/20 0.32
ALDH1A1 P00352 1/20 0.32
ALOX15 P16050 1/20 0.32
MRGPRX4 Q96LA9 1/20 0.32
RARB P10826 2/20 0.32
RARA P10276 1/20 0.32
RARG P13631 1/20 0.32
HMGB1 P09429 1/20 0.32
KEAP1 Q14145 1/20 0.32
NAPRT Q6XQN6 1/20 0.32
GSK3B P49841 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL974928 0.86 KDM4E (0.41) KDM4EASPHKDM8CYP1A2CES2
SCHEMBL27600988 0.84 KDM4E (0.35) KDM4EASPHKDM8CYP1A2ALDH1A1
SCHEMBL27912539 0.84 MRGPRX4 (0.46) FOLH1ALBALDH1A1ALOX15MRGPRX4
SCHEMBL9406148 0.81 RARB (0.41) KDM4EASPHKDM8CYP1A2CES2
SCHEMBL28785054 0.80 ALDH1A1 (0.40) KDM4ECES2CES1ALDH1A1MRGPRX4
SCHEMBL9419244 0.79 GABRP (0.46) RARBRARARARG
SCHEMBL5248959 0.79 GABRP (0.42) KDM4EASPHKDM8CYP1A2CES2
SCHEMBL542766 0.79 KDM4E (0.41) KDM4EASPHKDM8CYP1A2CES2
SCHEMBL9419332 0.77 RARB (0.51) ALOX15RARBRARARARG
SCHEMBL27985838 0.77 TSHR (0.46) KDM4EALDH1A1MRGPRX4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-104105691-A MODULATORS OF THE G PROTEIN-COUPLED MAS RECEPTOR AND THE TREATMENT OF DISORDERS RELATED THERETO ARENA PHARM INC 2014-10-15 CN disclosed