SCHEMBL28006116

SCHEMBL28006116

O=Cc1c[nH]c2ncc(Cl)nc12

nearest known ligand 0.40

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
KMT2A Q03164 1/20 0.40
MAPK1 P28482 3/20 0.34
CCNT1 O60563 1/20 0.32
CDK9 P50750 1/20 0.32
HASPIN Q8TF76 1/20 0.32
CYP2A6 P11509 1/20 0.30
IMPDH2 P12268 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL23830299 0.86 KMT2A (0.40) KMT2ACCNT1CDK9HASPINCYP2A6
SCHEMBL29936350 0.79 MAPK1 (0.57) KMT2AMAPK1CCNT1CDK9HASPIN
SCHEMBL12253387 0.79 KMT2A (0.40) KMT2AMAPK1CCNT1CDK9HASPIN
SCHEMBL1352440 0.79 MAPK1 (0.57) KMT2AMAPK1CCNT1CDK9HASPIN
SCHEMBL30259037 0.73 MAPK1 (0.62) MAPK1
SCHEMBL20846079 0.73 ALDH1A1 (0.41) MAPK1
SCHEMBL650607 0.73 MAPK1 (0.62) MAPK1
SCHEMBL1696892 0.72 KMT2A (0.55) KMT2AMAPK1CCNT1CDK9HASPIN
SCHEMBL14655319 0.71 JAK2 (0.40)
SCHEMBL15569859 0.71 KMT2A (0.36) KMT2ACCNT1CDK9HASPINCYP2A6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-104507945-A Pyrrolo[2,3-B]pyrazines as SYK inhibitors HOFFMANN LA ROCHE 2015-04-08 CN disclosed