SCHEMBL28006174

SCHEMBL28006174

COc1ncccc1C(=O)OI

nearest known ligand 0.53

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TDP1 Q9NUW8 1/20 0.53
L3MBTL1 Q9Y468 2/20 0.44
MAPT P10636 2/20 0.44
GAA P10253 2/20 0.44
SMN1; SMN2 Q16637 3/20 0.43
ALDH1A1 P00352 3/20 0.43
HTT P42858 1/20 0.43
MAPK1 P28482 2/20 0.42
SLC13A5 Q86YT5 1/20 0.42
NPC1 O15118 2/20 0.41
MEN1 O00255 1/20 0.41
TP53 P04637 1/20 0.41
RAB9A P51151 1/20 0.41
KMT2A Q03164 1/20 0.41
LMNA P02545 3/20 0.40
POLB P06746 1/20 0.40
HPGD P15428 1/20 0.40
MAP2K1 Q02750 1/20 0.40
BRD4 O60885 1/20 0.39
BRPF1 P55201 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL311206 0.86 TDP1 (0.69) TDP1L3MBTL1MAPTGAASMN1; SMN2
SCHEMBL28005008 0.83 TDP1 (0.53) TDP1L3MBTL1MAPTGAASMN1; SMN2
SCHEMBL28027851 0.83 TDP1 (0.53) TDP1L3MBTL1MAPTGAASMN1; SMN2
SCHEMBL949562 0.82 TDP1 (0.50) TDP1L3MBTL1MAPTGAASMN1; SMN2
SCHEMBL30592857 0.80 TDP1 (0.57) TDP1L3MBTL1MAPTGAASMN1; SMN2
SCHEMBL31081770 0.80 TDP1 (0.49) TDP1L3MBTL1MAPTGAASMN1; SMN2
SCHEMBL18201 0.80 TDP1 (0.57) TDP1L3MBTL1MAPTGAASMN1; SMN2
SCHEMBL8427582 0.80 TDP1 (0.49) TDP1L3MBTL1MAPTGAASMN1; SMN2
SCHEMBL9944383 0.80 MAPT (0.51) TDP1L3MBTL1MAPTGAASMN1; SMN2
SCHEMBL311599 0.80 L3MBTL1 (0.59) L3MBTL1MAPTSMN1; SMN2ALDH1A1HTT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-104507940-A Heterocyclic compounds TAKEDA PHARMACEUTICAL 2015-04-08 CN disclosed