SCHEMBL28006997

SCHEMBL28006997

O=C(O)C12CC3CC(C1)C(F)(F)C(C3)C2

nearest known ligand 0.41

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
L3MBTL1 Q9Y468 2/20 0.35
PKM P14618 1/20 0.35
HSD11B1 P28845 7/20 0.34
HTT P42858 2/20 0.34
KDM4E B2RXH2 1/20 0.34
ALDH1A1 P00352 2/20 0.33
HSD11B2 P80365 1/20 0.32
P2RX7 Q99572 1/20 0.32
CRHBP P24387 1/20 0.32
CRHR2 Q13324 1/20 0.32
MCOLN3 Q8TDD5 1/20 0.32
GLA P06280 1/20 0.32
THRB P10828 1/20 0.31
CYP2C9 P11712 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL25564585 0.80 HSD11B1 (0.32) L3MBTL1PKMHSD11B1HTTKDM4E
SCHEMBL12714 0.79 HSD11B1 (0.48) L3MBTL1PKMHSD11B1HTTKDM4E
SCHEMBL19557168 0.79 HSD11B1 (0.48) L3MBTL1PKMHSD11B1HTTKDM4E
SCHEMBL19557166 0.79 HSD11B1 (0.48) L3MBTL1PKMHSD11B1HTTKDM4E
SCHEMBL17041846 0.78 ALDH1A1 (0.32) L3MBTL1PKMALDH1A1
SCHEMBL12219710 0.78 ALDH1A1 (0.36) L3MBTL1PKMHSD11B1HTTKDM4E
SCHEMBL15827321 0.78 ALDH1A1 (0.36) L3MBTL1PKMHSD11B1HTTKDM4E
SCHEMBL17547624 0.77
SCHEMBL4389277 0.77 HSD11B1 (0.46) L3MBTL1PKMHSD11B1HTTKDM4E
SCHEMBL5489940 0.77 HSD11B1 (0.46) L3MBTL1PKMHSD11B1HTTKDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-104402883-B 4,4-difluoro diamantane carboxamides derivatives, pharmaceutical composition and its production and use Shanghai AQBioPharma Co. Ltd. (CN) 2016-04-27 CN disclosed
CN-104402883-A 4, 4-difluoroadamantane formamide derivative, pharmaceutical composition, preparation method and application thereof AIQIKANG MEDICAL TECHNOLOGY SHANGHAI CO LTD 2015-03-11 CN disclosed