SCHEMBL28008142

SCHEMBL28008142

CNS(=O)(=O)CCCOc1cc[c]c(CN)c1

nearest known ligand 0.38

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
PDIA6 Q15084 1/20 0.34
DUT P33316 1/20 0.32
ITGB3 P05106 1/20 0.31
ITGA2B P08514 1/20 0.31
CA12 O43570 1/20 0.31
CA1 P00915 1/20 0.31
CA2 P00918 1/20 0.31
TSHR P16473 1/20 0.31
CA7 P43166 1/20 0.31
CA9 Q16790 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9934246 0.87 KDM4E (0.32) PDIA6DUT
SCHEMBL28008529 0.85 FFAR1 (0.37) PDIA6CA12CA1CA2TSHR
SCHEMBL28008160 0.83 PDIA6 (0.37) PDIA6CA12CA1CA2TSHR
SCHEMBL9934856 0.82 PDIA6 (0.36) PDIA6DUT
SCHEMBL28008145 0.82 SYK (0.34) PDIA6CA12CA1CA2TSHR
SCHEMBL9935694 0.80
SCHEMBL28035468 0.79 ALDH1A1 (0.42) PDIA6
SCHEMBL27793390 0.77 TSHR (0.41) CA12CA1CA2TSHRCA7
SCHEMBL28008191 0.76 PDE3B (0.44)
SCHEMBL27999329 0.75 MAPT (0.39) CA12CA1CA2TSHRCA7

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-104710381-A Novel 3-hydroxy-5-arylisothiazole derivative MOCHIDA PHARM CO LTD 2015-06-17 CN disclosed
CN-102712610-B Novel 3-hydroxy-5-arylisothiazole derivatives MOCHIDA PHARM CO LTD 2015-03-04 CN disclosed