SCHEMBL28008449

SCHEMBL28008449

Cc1c(C(N)=O)ccc(-c2ccccn2)c1F

nearest known ligand 0.50

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
BTK Q06187 1/20 0.50
NPSR1 Q6W5P4 1/20 0.45
RXFP1 Q9HBX9 1/20 0.45
GRM5 P41594 2/20 0.44
SQOR Q9Y6N5 1/20 0.42
IKBKB O14920 1/20 0.42
KAT6A Q92794 2/20 0.40
MKNK1 Q9BUB5 1/20 0.38
MKNK2 Q9HBH9 1/20 0.38
CSNK1A1 P48729 1/20 0.38
TYRO3 Q06418 1/20 0.38
DYRK1B Q9Y463 1/20 0.38
TGFBR1 P36897 1/20 0.38
PARP1 P09874 1/20 0.38
DHODH Q02127 1/20 0.38
PARP2 Q9UGN5 1/20 0.38
CDC7 O00311 1/20 0.38
HCRTR1 O43613 2/20 0.38
HCRTR2 O43614 2/20 0.38
MAPT P10636 2/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2012719 0.81 GRM5 (0.53) BTKNPSR1RXFP1GRM5IKBKB
SCHEMBL22468488 0.79 BTK (0.46) BTKNPSR1RXFP1GRM5SQOR
SCHEMBL8815555 0.79 NPSR1 (0.47) BTKNPSR1RXFP1GRM5SQOR
SCHEMBL12828418 0.77 KDM4E (0.45) MAPTHTTBRD4LMNARAB9A
SCHEMBL22468497 0.77 BTK (0.58) BTKNPSR1RXFP1GRM5IKBKB
SCHEMBL29899091 0.77 GRM5 (0.49) BTKNPSR1RXFP1GRM5SQOR
SCHEMBL27491920 0.75 GRM5 (0.48) BTKNPSR1RXFP1GRM5SQOR
SCHEMBL997865 0.75 GRM5 (0.64) BTKNPSR1RXFP1GRM5CSNK1A1
SCHEMBL31249984 0.75 GRM5 (0.64) BTKNPSR1RXFP1GRM5CSNK1A1
SCHEMBL29506339 0.75 GRM5 (0.64) BTKNPSR1RXFP1GRM5CSNK1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-104540825-A Azaindolines HOFFMANN LA ROCHE 2015-04-22 CN disclosed