SCHEMBL28009074

SCHEMBL28009074

[c]1ncc(-n2cncn2)s1

nearest known ligand 0.38

Predicted protein targets (top 4)

geneUniProtsupporting neighboursconfidence
CYP2A6 P11509 1/20 0.38
KDM4E B2RXH2 1/20 0.34
ALDH1A1 P00352 1/20 0.34
SMN1; SMN2 Q16637 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL27903985 0.68 CYP2A6 (0.44) CYP2A6KDM4EALDH1A1SMN1; SMN2
Bromide SCHEMBL28124645 0.67 CYP2A6 (0.43) CYP2A6KDM4EALDH1A1SMN1; SMN2
SCHEMBL970243 0.65 CYP3A4 (0.39) CYP2A6ALDH1A1
SCHEMBL27954289 0.64 LMNA (0.38) CYP2A6KDM4EALDH1A1SMN1; SMN2
SCHEMBL18049511 0.61 KDM4E (0.34) CYP2A6KDM4EALDH1A1SMN1; SMN2
SCHEMBL27859244 0.61 CYP2A6 (0.61) CYP2A6KDM4EALDH1A1SMN1; SMN2
SCHEMBL14860938 0.60 CYP2A6 (0.37) CYP2A6KDM4EALDH1A1SMN1; SMN2
SCHEMBL27905069 0.60 SMN1; SMN2 (0.72) CYP2A6KDM4EALDH1A1SMN1; SMN2
SCHEMBL18327504 0.58 KDM4E (0.35) CYP2A6KDM4EALDH1A1SMN1; SMN2
SCHEMBL9078549 0.58

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-105503850-B N [base of 4 tert-butyl group 5 (base of 1,2,4 triazole 1) thiazole 2] lauramides and its application 湖南大学 2018-01-09 CN disclosed
CN-104876924-B 3 [base] benzoxazinones of 5 (base of 1,2,4 triazole 1) thiazole 2 and preparation method and application 湖南大学 2017-06-23 CN disclosed
CN-105503850-A N-[5-(1,2,4-triazol-1-yl)thiazol-2-yl]lauramide and application thereof UNIV HUNAN 2016-04-20 CN disclosed
CN-103664928-B N- [5- (1,2, 4-triazol-1-yl) thiazol-2-yl ] fatty amide and application thereof HUNAN UNIVERSITY (CN) 2015-10-07 CN disclosed
CN-103664927-B N-[5-(1,2,4-triazole-1-yl)thiazole-2-yl]aryl amide, preparation method, and applications thereof UNIV HUNAN 2015-06-24 CN disclosed
CN-104628716-A N-[5-(1,2,4-triazolyl-1-yl)thiazolyl-2-yl]lauramide and application thereof UNIV HUNAN 2015-05-20 CN disclosed